日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Oral obeldesivir provides postexposure protection against Marburg virus in nonhuman primates

口服奥贝地西韦可为非人灵长类动物提供暴露后针对马尔堡病毒的保护作用

Cross, Robert W; Woolsey, Courtney; Prasad, Abhishek N; Borisevich, Viktoriya; Agans, Krystle N; Deer, Daniel J; Harrison, Mack B; Dobias, Natalie S; Fenton, Karla A; Cihlar, Tomas; Nguyen, Anh-Quan; Babusis, Darius; Bannister, Roy; Vermillion, Meghan S; Chu, Victor C; Geisbert, Thomas W

The oral drug obeldesivir protects nonhuman primates against lethal Ebola virus infection.

口服药物奥贝尔地西韦可保护非人灵长类动物免受致命的埃博拉病毒感染

Woolsey Courtney, Cross Robert W, Chu Victor C, Prasad Abhishek N, Agans Krystle N, Borisevich Viktoriya, Deer Daniel J, Harrison Mack B, Martinez Jasmine K, Dobias Natalie S, Fenton Karla A, Cihlar Tomas, Nguyen Anh-Quan, Babusis Darius, Bannister Roy, Vermillion Meghan S, Geisbert Thomas W

A Randomized, Blinded, Vehicle-Controlled Dose-Ranging Study to Evaluate and Characterize Remdesivir Efficacy Against Ebola Virus in Rhesus Macaques

一项随机、双盲、载体对照剂量范围研究,旨在评估和表征瑞德西韦对恒河猴埃博拉病毒的疗效

Zumbrun, Elizabeth E; Garvey, Carly B; Wells, Jay B; Lynn, Ginger C; Van Tongeren, Sean A; Steffens, Jesse T; Wetzel, Kelly S; Wetzel, Darrell L; Esham, Heather L; Garza, Nicole L; Lee, Eric D; Scruggs, Jennifer L; Rossi, Franco D; Brown, Elizabeth S; Weidner, Jessica M; Gomba, Laura M; O'Brien, Kristan A; Jay, Alexandra N; Zeng, Xiankun; Akers, Kristen S; Kallgren, Paul A; Englund, Ethan; Meinig, J Matthew; Kugelman, Jeffrey R; Moore, Joshua L; Bloomfield, Holly A; Norris, Sarah L; Bryan, Tameka; Scheuerell, Christie H; Walters, Jesse; Mollova, Nevena; Blair, Christiana; Babusis, Darius; Cihlar, Tomas; Porter, Danielle P; Singh, Bali; Hedskog, Charlotte; Bavari, Sina; Warren, Travis K; Bannister, Roy

Characterization of the Cynomolgus Macaque Model of Marburg Virus Disease and Assessment of Timing for Therapeutic Treatment Testing

食蟹猴马尔堡病毒病模型的特征分析及治疗试验时机的评估

Zumbrun, Elizabeth E; Garvey, Carly B; Wells, Jay B; Lynn, Ginger C; Van Tongeren, Sean; Steffens, Jesse T; Wetzel, Kelly S; Gomba, Laura M; O'Brien, Kristan A; Rossi, Franco D; Zeng, Xiankun; Lee, Eric D; Raymond, Jo Lynne W; Hoffman, Diana A; Jay, Alexandra N; Brown, Elizabeth S; Kallgren, Paul A; Norris, Sarah L; Cantey-Kiser, Jean; Kudiya, Humza; Arthur, Chris; Blair, Christiana; Babusis, Darius; Chu, Victor C; Singh, Bali; Bannister, Roy; Porter, Danielle P; Cihlar, Tomas; Dye, John M

Efficacy of the oral nucleoside prodrug GS-5245 (Obeldesivir) against SARS-CoV-2 and coronaviruses with pandemic potential

口服核苷前药GS-5245(奥贝地西韦)对SARS-CoV-2和具有大流行潜力的冠状病毒的疗效

Martinez, David R; Moreira, Fernando R; Zweigart, Mark R; Gully, Kendra L; De la Cruz, Gabriela; Brown, Ariane J; Adams, Lily E; Catanzaro, Nicholas; Yount, Boyd; Baric, Thomas J; Mallory, Michael L; Conrad, Helen; May, Samantha R; Dong, Stephanie; Scobey, D Trevor; Montgomery, Stephanie A; Perry, Jason; Babusis, Darius; Barrett, Kimberly T; Nguyen, Anh-Hoa; Nguyen, Anh-Quan; Kalla, Rao; Bannister, Roy; Bilello, John P; Feng, Joy Y; Cihlar, Tomas; Baric, Ralph S; Mackman, Richard L; Schäfer, Alexandra; Sheahan, Timothy P

Nucleotide Prodrug Containing a Nonproteinogenic Amino Acid To Improve Oral Delivery of a Hepatitis C Virus Treatment

含有非蛋白源性氨基酸的核苷酸前药可改善丙型肝炎病毒治疗药物的口服递送

Feng, Joy Y; Wang, Ting; Park, Yeojin; Babusis, Darius; Birkus, Gabriel; Xu, Yili; Voitenleitner, Christian; Fenaux, Martijn; Yang, Huiling; Eng, Stacey; Tirunagari, Neeraj; Kirschberg, Thorsten; Cho, Aesop; Ray, Adrian S

Sofosbuvir and Ribavirin Liver Pharmacokinetics in Patients Infected with Hepatitis C Virus

丙型肝炎病毒感染患者体内索非布韦和利巴韦林的肝脏药代动力学

Babusis, Darius; Curry, Michael P; Kirby, Brian; Park, Yeojin; Murakami, Eisuke; Wang, Ting; Mathias, Anita; Afdhal, Nezam; McHutchison, John G; Ray, Adrian S

Broad-spectrum antiviral GS-5734 inhibits both epidemic and zoonotic coronaviruses

广谱抗病毒药物GS-5734可抑制流行性冠状病毒和人畜共患冠状病毒。

Sheahan, Timothy P; Sims, Amy C; Graham, Rachel L; Menachery, Vineet D; Gralinski, Lisa E; Case, James B; Leist, Sarah R; Pyrc, Krzysztof; Feng, Joy Y; Trantcheva, Iva; Bannister, Roy; Park, Yeojin; Babusis, Darius; Clarke, Michael O; Mackman, Richard L; Spahn, Jamie E; Palmiotti, Christopher A; Siegel, Dustin; Ray, Adrian S; Cihlar, Tomas; Jordan, Robert; Denison, Mark R; Baric, Ralph S

Viability of primary osteoblasts after treatment with tenofovir alafenamide: Lack of cytotoxicity at clinically relevant drug concentrations

替诺福韦艾拉酚胺治疗后原代成骨细胞的存活率:在临床相关药物浓度下无细胞毒性

Callebaut, Christian; Liu, Yang; Babusis, Darius; Ray, Adrian; Miller, Michael; Kitrinos, Kathryn

Implications of efficient hepatic delivery by tenofovir alafenamide (GS-7340) for hepatitis B virus therapy

替诺福韦艾拉酚胺(GS-7340)高效肝脏递送对乙型肝炎病毒治疗的意义

Murakami, Eisuke; Wang, Ting; Park, Yeojin; Hao, Jia; Lepist, Eve-Irene; Babusis, Darius; Ray, Adrian S