日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Biological Activity and Structural Biology of Current KAT6A Inhibitor Chemotypes.

当前KAT6A抑制剂化学类型的生物活性和结构生物学。

Suwandi Adi, Jin Jianwen, Zhao Yichao, Mudududdla Ramesh, Gee Yi Sing, Deora Girdhar Singh, Sun Yuxin, Wei Heping, Huang Fei, He Jin-Shu, George Amee J, Hermans Stefan J, Leaver David J, Parker Michael W, Baell Jonathan B

Fluorinated pyrimidine 5-carboxamides as potential tools for MERTK targeted fluorine-18-PET-radioligand development

氟化嘧啶5-甲酰胺作为MERTK靶向氟-18-PET放射性配体开发的潜在工具

Mudududdla, Ramesh; Wong, Siu Wai; Nguyen, Nghi; Xue, Lian; Stashko, Michael A; Wang, Xiaodong; Vivash, Lucy; Binder, Michele D; Ackermann, Uwe; Bozikis, Ylva E; Kilpatrick, Trevor J; Baell, Jonathan B

Heterocyclic core modifications in trypanosomacidal 2-[(phenylheteroaryl)ethyl]ureas

锥虫杀灭剂 2-[(苯基杂芳基)乙基]脲的杂环核心修饰

Toynton, Arthur; Ferrins, Lori; Newson, Harriet L; Sykes, Melissa L; Varghese, Swapna; Nguyen, Nghi; Russell, Stephanie; Rahmani, Raphaël; Cheang, Jeremy; Flematti, Gavin R; Skelton, Brian W; Zulfiqar, Bilal; Avery, Vicky M; Baell, Jonathan B; Piggott, Matthew J

A Collection of Useful Nuisance Compounds (CONS) for Interrogation of Bioassay Integrity

用于检测生物测定完整性的有用干扰化合物 (CONS) 集合

Hu, Huabin; Yi, Xiangyan; Xue, Lian; Baell, Jonathan B

Visible-light-induced N-alkylation of anilines with 4-hydroxybutan-2-one

可见光诱导的苯胺与4-羟基丁-2-酮的N-烷基化反应

Jiang, Liya; Ni, Ling; Tang, Xinyue; Baell, Jonathan B; Huang, Fei; Ren, Lanhui

Novel Diacyl-hydrazide Compounds as Potential Therapeutics for Visceral Leishmaniasis

新型二酰肼化合物作为内脏利什曼病的潜在治疗药物

Bernhard Jandl, Rebecca Zheng, Markus Muttenthaler, Jonathan Baell

Phenotypic-Based Discovery and Exploration of a Resorufin Scaffold with Activity against Mycobacterium tuberculosis

基于表型的发现和探索具有抗结核分枝杆菌活性的试卤灵骨架

Tran, Eric; Cheung, Chen-Yi; Li, Lucy; Carter, Glen P; Gable, Robert W; West, Nicholas P; Kaur, Amandeep; Gee, Yi Sing; Cook, Gregory M; Baell, Jonathan B; Jörg, Manuela

A MOZ-TIF2 leukemia mouse model displays KAT6-dependent H3K23 propionylation and overexpression of a set of active developmental genes

MOZ-TIF2 白血病小鼠模型表现出 KAT6 依赖的 H3K23 丙酰化和一组活跃发育基因的过度表达

Anne E Smolko, Daniel W Sullivan, Sarah Naomi Olsen, Hyuckjoon Kang, Samuel D Whedon, Jonathan B Baell, Philip A Cole, Scott A Armstrong, Mitzi I Kuroda

A small molecule inhibitor of PTP1B and PTPN2 enhances T cell anti-tumor immunity

PTP1B 和 PTPN2 的小分子抑制剂可增强 T 细胞抗肿瘤免疫力。

Shuwei Liang # ,Eric Tran # ,Xin Du ,Jiajun Dong ,Harrison Sudholz ,Hao Chen ,Zihan Qu ,Nicholas D Huntington ,Jeffrey J Babon ,Nadia J Kershaw ,Zhong-Yin Zhang ,Jonathan B Baell ,Florian Wiede ,Tony Tiganis

Novel Perspectives on the Design and Development of a Long-Acting Subcutaneous Raltegravir Injection for Treatment of HIV-In Vitro and In Vivo Evaluation

治疗艾滋病毒的长效皮下雷替拉韦注射剂的设计和开发新视角-体外和体内评价

Heba S Abd-Ellah, Ramesh Mudududdla, Glen P Carter, Jonathan B Baell