Design of Selective PAK1 Inhibitor G-5555: Improving Properties by Employing an Unorthodox Low-pK a Polar Moiety
选择性 PAK1 抑制剂 G-5555 的设计:通过采用非传统低 pK 极性部分来改善性能
期刊:ACS Medicinal Chemistry Letters
影响因子:3.5
doi:10.1021/acsmedchemlett.5b00398
Chudi O Ndubaku, James J Crawford, Joy Drobnick, Ignacio Aliagas, David Campbell, Ping Dong, Laura M Dornan, Sergio Duron, Jennifer Epler, Lewis Gazzard, Christopher E Heise, Klaus P Hoeflich, Diana Jakubiak, Hank La, Wendy Lee, Baiwei Lin, Joseph P Lyssikatos, Jasna Maksimoska, Ronen Marmorstein, L