日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Rescue of autoimmune hepatitis by soluble MHC class II molecules in an altered concanavalin A-induced experimental model

可溶性 MHC II 类分子在改变的刀豆球蛋白 A 诱发的实验模型中挽救自身免疫性肝炎

Katerina Bakela, Maria Georgia Dimitraki, Evangelia Skoufa, Irene Athanassakis

Soluble major histocompatibility complex molecules in immune regulation: highlighting class II antigens

可溶性主要组织相容性复合体分子在免疫调节中的作用:重点关注II类抗原

Bakela, Katerina; Athanassakis, Irene

Identification of a 4-fluorobenzyl l-valinate amide benzoxaborole (AN11736) as a potential development candidate for the treatment of Animal African Trypanosomiasis (AAT)

鉴定出一种 4-氟苄基 L-缬氨酸酰胺苯并硼氧杂环戊烯 (AN11736) 作为治疗动物非洲锥虫病 (AAT) 的潜在候选药物

Akama, Tsutomu; Zhang, Yong-Kang; Freund, Yvonne R; Berry, Pamela; Lee, Joanne; Easom, Eric E; Jacobs, Robert T; Plattner, Jacob J; Witty, Michael J; Peter, Rosemary; Rowan, Tim G; Gillingwater, Kirsten; Brun, Reto; Nare, Bakela; Mercer, Luke; Xu, Musheng; Wang, Jiangong; Liang, Hao

Synergy between dinotefuran and fipronil against the cat flea (Ctenocephalides felis): improved onset of action and residual speed of kill in adult cats

呋虫胺和氟虫腈对猫蚤(Ctenocephalides felis)具有协同作用:可提高成年猫的起效速度和残留杀灭率。

Delcombel, Romain; Karembe, Hamadi; Nare, Bakela; Burton, Audrey; Liebenberg, Julian; Fourie, Josephus; Varloud, Marie

Open Source Drug Discovery with the Malaria Box Compound Collection for Neglected Diseases and Beyond

利用疟疾化合物库进行开源药物发现,以应对被忽视的热带病及其他疾病

Van Voorhis, Wesley C; Adams, John H; Adelfio, Roberto; Ahyong, Vida; Akabas, Myles H; Alano, Pietro; Alday, Aintzane; Alemán Resto, Yesmalie; Alsibaee, Aishah; Alzualde, Ainhoa; Andrews, Katherine T; Avery, Simon V; Avery, Vicky M; Ayong, Lawrence; Baker, Mark; Baker, Stephen; Ben Mamoun, Choukri; Bhatia, Sangeeta; Bickle, Quentin; Bounaadja, Lotfi; Bowling, Tana; Bosch, Jürgen; Boucher, Lauren E; Boyom, Fabrice F; Brea, Jose; Brennan, Marian; Burton, Audrey; Caffrey, Conor R; Camarda, Grazia; Carrasquilla, Manuela; Carter, Dee; Belen Cassera, Maria; Chih-Chien Cheng, Ken; Chindaudomsate, Worathad; Chubb, Anthony; Colon, Beatrice L; Colón-López, Daisy D; Corbett, Yolanda; Crowther, Gregory J; Cowan, Noemi; D'Alessandro, Sarah; Le Dang, Na; Delves, Michael; DeRisi, Joseph L; Du, Alan Y; Duffy, Sandra; Abd El-Salam El-Sayed, Shimaa; Ferdig, Michael T; Fernández Robledo, José A; Fidock, David A; Florent, Isabelle; Fokou, Patrick V T; Galstian, Ani; Gamo, Francisco Javier; Gokool, Suzanne; Gold, Ben; Golub, Todd; Goldgof, Gregory M; Guha, Rajarshi; Guiguemde, W Armand; Gural, Nil; Guy, R Kiplin; Hansen, Michael A E; Hanson, Kirsten K; Hemphill, Andrew; Hooft van Huijsduijnen, Rob; Horii, Takaaki; Horrocks, Paul; Hughes, Tyler B; Huston, Christopher; Igarashi, Ikuo; Ingram-Sieber, Katrin; Itoe, Maurice A; Jadhav, Ajit; Naranuntarat Jensen, Amornrat; Jensen, Laran T; Jiang, Rays H Y; Kaiser, Annette; Keiser, Jennifer; Ketas, Thomas; Kicka, Sebastien; Kim, Sunyoung; Kirk, Kiaran; Kumar, Vidya P; Kyle, Dennis E; Lafuente, Maria Jose; Landfear, Scott; Lee, Nathan; Lee, Sukjun; Lehane, Adele M; Li, Fengwu; Little, David; Liu, Liqiong; Llinás, Manuel; Loza, Maria I; Lubar, Aristea; Lucantoni, Leonardo; Lucet, Isabelle; Maes, Louis; Mancama, Dalu; Mansour, Nuha R; March, Sandra; McGowan, Sheena; Medina Vera, Iset; Meister, Stephan; Mercer, Luke; Mestres, Jordi; Mfopa, Alvine N; Misra, Raj N; Moon, Seunghyun; Moore, John P; Morais Rodrigues da Costa, Francielly; Müller, Joachim; Muriana, Arantza; Nakazawa Hewitt, Stephen; Nare, Bakela; Nathan, Carl; Narraidoo, Nathalie; Nawaratna, Sujeevi; Ojo, Kayode K; Ortiz, Diana; Panic, Gordana; Papadatos, George; Parapini, Silvia; Patra, Kailash; Pham, Ngoc; Prats, Sarah; Plouffe, David M; Poulsen, Sally-Ann; Pradhan, Anupam; Quevedo, Celia; Quinn, Ronald J; Rice, Christopher A; Abdo Rizk, Mohamed; Ruecker, Andrea; St Onge, Robert; Salgado Ferreira, Rafaela; Samra, Jasmeet; Robinett, Natalie G; Schlecht, Ulrich; Schmitt, Marjorie; Silva Villela, Filipe; Silvestrini, Francesco; Sinden, Robert; Smith, Dennis A; Soldati, Thierry; Spitzmüller, Andreas; Stamm, Serge Maximilian; Sullivan, David J; Sullivan, William; Suresh, Sundari; Suzuki, Brian M; Suzuki, Yo; Swamidass, S Joshua; Taramelli, Donatella; Tchokouaha, Lauve R Y; Theron, Anjo; Thomas, David; Tonissen, Kathryn F; Townson, Simon; Tripathi, Abhai K; Trofimov, Valentin; Udenze, Kenneth O; Ullah, Imran; Vallieres, Cindy; Vigil, Edgar; Vinetz, Joseph M; Voong Vinh, Phat; Vu, Hoan; Watanabe, Nao-Aki; Weatherby, Kate; White, Pamela M; Wilks, Andrew F; Winzeler, Elizabeth A; Wojcik, Edward; Wree, Melanie; Wu, Wesley; Yokoyama, Naoaki; Zollo, Paul H A; Abla, Nada; Blasco, Benjamin; Burrows, Jeremy; Laleu, Benoît; Leroy, Didier; Spangenberg, Thomas; Wells, Timothy; Willis, Paul A

Soluble MHC-II proteins promote suppressive activity in CD4+ T cells

可溶性 MHC-II 蛋白促进 CD4+ T 细胞的抑制活性

Katerina Bakela, Nikos Kountourakis, Michalis Aivaliotis, Irene Athanassakis

Targeting Lysine Deacetylases (KDACs) in Parasites

靶向寄生虫中的赖氨酸脱乙酰酶(KDACs)

Wang, Qi; Rosa, Bruce A; Nare, Bakela; Powell, Kerrie; Valente, Sergio; Rotili, Dante; Mai, Antonello; Marshall, Garland R; Mitreva, Makedonka

Pharmacokinetics and pharmacodynamics utilizing unbound target tissue exposure as part of a disposition-based rationale for lead optimization of benzoxaboroles in the treatment of Stage 2 Human African Trypanosomiasis

利用游离靶组织暴露量作为基于处置原理的苯并硼氧杂环化合物先导化合物优化方法,研究其在治疗第二阶段人类非洲锥虫病中的药代动力学和药效学。

Wring, Stephen; Gaukel, Eric; Nare, Bakela; Jacobs, Robert; Beaudet, Beth; Bowling, Tana; Mercer, Luke; Bacchi, Cyrus; Yarlett, Nigel; Randolph, Ryan; Parham, Robin; Rewerts, Cindy; Platner, Jacob; Don, Robert

SCYX-7158, an orally-active benzoxaborole for the treatment of stage 2 human African trypanosomiasis

SCYX-7158,一种口服有效的苯并硼氧杂环化合物,用于治疗2期人类非洲锥虫病

Jacobs, Robert T; Nare, Bakela; Wring, Stephen A; Orr, Matthew D; Chen, Daitao; Sligar, Jessica M; Jenks, Matthew X; Noe, Robert A; Bowling, Tana S; Mercer, Luke T; Rewerts, Cindy; Gaukel, Eric; Owens, Jennifer; Parham, Robin; Randolph, Ryan; Beaudet, Beth; Bacchi, Cyrus J; Yarlett, Nigel; Plattner, Jacob J; Freund, Yvonne; Ding, Charles; Akama, Tsutomu; Zhang, Y-K; Brun, Reto; Kaiser, Marcel; Scandale, Ivan; Don, Robert

2,4-Diaminopyrimidines as potent inhibitors of Trypanosoma brucei and identification of molecular targets by a chemical proteomics approach

2,4-二氨基嘧啶作为布氏锥虫的有效抑制剂以及通过化学蛋白质组学方法识别分子靶点

Luke Mercer, Tana Bowling, Joe Perales, Jennifer Freeman, Tien Nguyen, Cyrus Bacchi, Nigel Yarlett, Robert Don, Robert Jacobs, Bakela Nare