日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Biologics developability data analysis using hierarchical clustering accelerates candidate lead selection, optimization, and preformulation screening.

利用层次聚类进行生物制剂可开发性数据分析,可以加速候选先导化合物的选择、优化和制剂前筛选

Metcalf Kevin James, Wo Galen, Zaragoza Jan Paulo, Raoufi Fahimeh, Baker Jeanne, Chen Daoyang, Derebe Mehabaw, Hogan Jason, Hsu Amy, Kofman Esther, Leigh David, Li Mandy, Malashock Dan, Mann Cate, Motlagh Soha, Park Jihea, Sathiyamoorthy Karthik, Shidhore Madhura, Tang Yinyan, Teng Kevin, Williams Katharine, Waight Andrew, Yilmaz Sultan, Zhang Fan, Zhong Huimin, Fayadat-Dilman Laurence, Bailly Marc

Preclinical development of MK‐2214 a novel antibody targeting pS413 tau for the treatment of Alzheimer’s Disease

MK-2214是一种靶向pS413 tau的新型抗体,目前正处于治疗阿尔茨海默病的临床前开发阶段。

Elmore, Susan A; Berridge, Brian R; Boyle, Michael C; Cora, Michelle C; Hoenerhoff, Mark J; Kooistra, Linda; Laast, Victoria A; Morrison, James P; Rao, Deepa; Rinke, Matthias; Yoshizawa, Katsuhiko; Sugam, Jonathan A; Robey, Seth; Suon, Sokreine; Tian, Yuan; Wong, Oitak; Zhao, Xuemei; Chen, Ying; Judo, Michael; Smith, Brad E; Popescu, Andrei; Kurz, Jonathan; Herring, W Joseph; Baker, Jeanne; Parmentier‐Batteur, Sophie; Klein, Rebecca M; Smith, Sean M; Uslaner, Jason M

Amyloid precursor protein selective gamma-secretase inhibitors for treatment of Alzheimer's disease.

用于治疗阿尔茨海默病的淀粉样前体蛋白选择性γ-分泌酶抑制剂

Basi Guriqbal S, Hemphill Susanna, Brigham Elizabeth F, Liao Anna, Aubele Danielle L, Baker Jeanne, Barbour Robin, Bova Michael, Chen Xiao-Hua, Dappen Michael S, Eichenbaum Tovah, Goldbach Erich, Hawkinson Jon, Lawler-Herbold Rose, Hu Kang, Hui Terence, Jagodzinski Jacek J, Keim Pamela S, Kholodenko Dora, Latimer Lee H, Lee Mike, Marugg Jennifer, Mattson Matthew N, McCauley Scott, Miller James L, Motter Ruth, Mutter Linda, Neitzel Martin L, Ni Huifang, Nguyen Lan, Quinn Kevin, Ruslim Lany, Semko Christopher M, Shapiro Paul, Smith Jenifer, Soriano Ferdie, Szoke Balazs, Tanaka Kevin, Tang Pearl, Tucker John A, Ye Xiacong Michael, Yu Mei, Wu Jing, Xu Ying-Zi, Garofalo Albert W, Sauer John Michael, Konradi Andrei W, Ness Daniel, Shopp George, Pleiss Michael A, Freedman Stephen B, Schenk Dale