The Dysregulated Pharmacology of Clinically Relevant ESR1 Mutants is Normalized by Ligand-activated WT Receptor.
临床相关 ESR1 突变体的药理学失调可通过配体激活的野生型受体恢复正常
期刊:Molecular Cancer Therapeutics
影响因子:5.5
doi:10.1158/1535-7163.MCT-19-1148
Andreano Kaitlyn J, Baker Jennifer G, Park Sunghee, Safi Rachid, Artham Sandeep, Oesterreich Steffi, Jeselsohn Rinath, Brown Myles, Sammons Sarah, Wardell Suzanne E, Chang Ching-Yi, Norris John D, McDonnell Donald P