日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Histone methyltransferase PRDM9 promotes survival of drug-tolerant persister cells in glioblastoma.

组蛋白甲基转移酶PRDM9促进胶质母细胞瘤中耐药持续细胞的存活。

Joun George L, Kempe Emma G, Chen Brianna, Sterling Jayden R, Abbassi Ramzi H, Friess Dana, Singleton Matthew, Choudhury Chandra, Marian Oana C, du Preez W Daniel, Recasens Ariadna, Clark Teleri, Du Tian Y, Low Jason K K, Kim Hani, Yang Pengyi, Khor Jasmine, Hoque Monira, Indurthi Dinesh C, Kuchibhotla Mani, Palanisamy Ranjith, Jorgensen William T, Montgomery Andrew P, Baker Jennifer R, Higginbottom Sarah L, Tomaskovic-Crook Eva, Crook Jeremy M, Loo Lipin, Day Bryan W, Neely G Gregory, Guccione Ernesto, Johns Terrance G, Kassiou Michael, Feng Yuchen, Harris Lachlan, Don Anthony S, Munoz Lenka

Exploration of hydrazine-based small molecules as metal chelators for KDM4 inhibition.

探索肼类小分子作为金属螯合剂抑制KDM4

Saxton Angus J, Sterling Jayden, Hamilton Michael P, Abbassi Ramzi H, McCluskey Adam, Munoz Lenka, Baker Jennifer R

Cryo-EM Reveals Regulatory Mechanisms Governing Substrate Selection and Activation of Human LONP1

冷冻电镜揭示了调控人 LONP1 底物选择和激活的机制

Mindrebo, Jeffrey T; Alexandrescu, Lauren; Baker, Jennifer R; Wang, Garret; Lander, Gabriel C

Next-generation of BBQ analogues that selectively target breast cancer

下一代选择性靶向乳腺癌的烧烤类似物

Baker, Jennifer R; Gilbert, Jayne; O'Brien, Nicholas S; Russell, Cecilia C; McCluskey, Adam; Sakoff, Jennette A

Systematic literature review reveals suboptimal use of chemical probes in cell-based biomedical research

系统性文献综述揭示了化学探针在基于细胞的生物医学研究中的不合理使用。

Sterling, Jayden; Baker, Jennifer R; McCluskey, Adam; Munoz, Lenka

Amino Alcohols as Potential Antibiotic and Antifungal Leads.

氨基醇作为潜在的抗生素和抗真菌先导化合物

Baker Jennifer R, Cossar Peter J, Blaskovich Mark A T, Elliott Alysha G, Zuegg Johannes, Cooper Matthew A, Lewis Peter J, McCluskey Adam

Light-mediated multi-target protein degradation using arylazopyrazole photoswitchable PROTACs (AP-PROTACs)

利用芳基偶氮吡唑光开关PROTACs(AP-PROTACs)进行光介导的多靶点蛋白降解

Zhang, Qisi; Kounde, Cyrille S; Mondal, Milon; Greenfield, Jake L; Baker, Jennifer R; Kotelnikov, Sergei; Ignatov, Mikhail; Tinworth, Christopher P; Zhang, Leran; Conole, Daniel; De Vita, Elena; Kozakov, Dima; McCluskey, Adam; Harling, John D; Fuchter, Matthew J; Tate, Edward W

Antigiardial Activity of Novel Guanidine Compounds

新型胍类化合物的抗贾第鞭毛虫活性

Stevens, Andrew J; Abraham, Rebecca; Young, Kelly A; Russell, Cecilia C; McCluskey, Siobhann N; Baker, Jennifer R; Rusdi, Bertha; Page, Stephen W; O'Handley, Ryan; O'Dea, Mark; Abraham, Sam; McCluskey, Adam

Discovery of 4,6-bis(2-((E)-benzylidene)hydrazinyl)pyrimidin-2-Amine with Antibiotic Activity

发现具有抗生素活性的4,6-双(2-((E)-亚苄基)肼基)嘧啶-2-胺

Russell, Cecilia C; Stevens, Andrew; Young, Kelly A; Baker, Jennifer R; McCluskey, Siobhann N; Khazandi, Manouchehr; Pi, Hongfei; Ogunniyi, Abiodun; Page, Stephen W; Trott, Darren J; McCluskey, Adam

Disulfiram effects on responses to intravenous cocaine administration

双硫仑对静脉注射可卡因反应的影响

Baker, Jennifer R; Jatlow, Peter; McCance-Katz, Elinore F