Optimization of Physicochemical Properties and ADME for 2,4-Substituted 1H-Pyrrolo[2,3b]pyridines Inhibitors of Trypanosome Proliferation
2,4-取代的1H-吡咯并[2,3b]吡啶类锥虫增殖抑制剂的理化性质和ADME优化
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c01217
Bachovchin, Kelly A; Díaz, Rosario; Ceballos-Perez, Gloria; Rojas-Barros, Domingo; Pérez-Moreno, Guiomar; García-Hernández, Raquel; Bosch-Navarrete, Cristina; Rivers, Mitch; Penn, Erica C; Roncal, Norma E; Sciotti, Richard J; Campbell, Robert F; Martinez-Martinez, Maria Santos; Manzano-Chinchon, Pilar; Ruiz-Perez, Luis Miguel; Navarro, Miguel; González-Pacanowska, Dolores; Pollastri, Michael P; Ferrins, Lori; Singh, Baljinder