日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Novel NPY2R agonist BI 1820237 provides synergistic anti-obesity efficacy when combined with the GCGR/GLP-1R dual agonist survodutide

新型NPY2R激动剂BI 1820237与GCGR/GLP-1R双重激动剂苏沃度肽联合使用时,可产生协同抗肥胖疗效。

Augustin, Robert; Oldenburger, Anouk; Baader-Pagler, Tamara; Zimmermann, Tina; Borghardt, Jens; Hecksher-Sørensen, Jacob; Baljuls, Angela; Reindl, Wolfgang; Krawczyk, Bartlomiej; Martel, Eric; Brennauer, Albert; Peters, Stefan; Grube, Achim; Rudkjaer, Lise Biehl; Haebel, Peter

Effects of a long-acting secretin peptide analog alone and in combination with a GLP-1R agonist in a diet-induced obesity mouse model

长效促胰液素肽类似物单独使用和与 GLP-1R 激动剂联合使用对饮食诱导的肥胖小鼠模型的影响

Mona Loeffler, Katarina Klepac, Angela Baljuls, Bradford Hamilton, Svenja Mayer-Wrangowski, Peter Haebel, Tina Zimmermann

GPR101 loss promotes insulin resistance and diet-induced obesity risk.

GPR101 缺失会促进胰岛素抵抗和饮食诱导的肥胖风险

Garrett Lillian, Irmler Martin, Baljuls Angela, Rathkolb Birgit, Dragano Nathalia, Gerlini Raffaele, Sanz-Moreno Adrián, Aguilar-Pimentel Antonio, Becker Lore, Kraiger Markus, Reithmeir Rosa, Beckers Johannes, Calzada-Wack Julia, Wurst Wolfgang, Fuchs Helmut, Gailus-Durner Valerie, Zimmermann Tina, Hölter Sabine M, de Angelis Martin Hrabě

The calcitonin receptor is the main mediator of LAAMA's body weight lowering effects in male mice

降钙素受体是 LAAMA 对雄性小鼠产生减重作用的主要介质

Salome Gamakharia, Christelle Le Foll, Wolfgang Rist, Tamara Baader-Pagler, Angela Baljuls, Thomas A Lutz

Tyr728 in the kinase domain of the murine kinase suppressor of RAS 1 regulates binding and activation of the mitogen-activated protein kinase kinase

RAS 1 小鼠激酶抑制因子激酶结构域中的 Tyr728 可调节丝裂原活化蛋白激酶激酶的结合和活化

Claudia Sibilski, Thomas Mueller, Laxmikanth Kollipara, René P Zahedi, Ulf R Rapp, Thomas Rudel, Angela Baljuls

Raf kinases mediate the phosphorylation of eukaryotic translation elongation factor 1A and regulate its stability in eukaryotic cells

Raf激酶介导真核翻译延伸因子1A的磷酸化,并调节其在真核细胞中的稳定性。

Sanges, C; Scheuermann, C; Zahedi, R P; Sickmann, A; Lamberti, A; Migliaccio, N; Baljuls, A; Marra, M; Zappavigna, S; Reinders, J; Rapp, U; Abbruzzese, A; Caraglia, M; Arcari, P

The tumor suppressor DiRas3 forms a complex with H-Ras and C-RAF proteins and regulates localization, dimerization, and kinase activity of C-RAF

肿瘤抑制因子 DiRas3 与 H-Ras 和 C-RAF 蛋白形成复合物,并调节 C-RAF 的定位、二聚化和激酶活性

Angela Baljuls, Matthias Beck, Ayla Oenel, Armin Robubi, Ruth Kroschewski, Mirko Hekman, Thomas Rudel, Ulf R Rapp

BAD contributes to RAF-mediated proliferation and cooperates with B-RAF-V600E in cancer signaling

BAD 促进 RAF 介导的增殖,并与 B-RAF-V600E 协同作用,促进癌症信号传导

Lisa Polzien, Angela Baljuls, Marco Albrecht, Mirko Hekman, Ulf R Rapp

Impaired binding of 14-3-3 to C-RAF in Noonan syndrome suggests new approaches in diseases with increased Ras signaling

努南综合征中 14-3-3 与 C-RAF 结合受损提示,应采取新方法治疗 Ras 信号传导增强的疾病

Manuela Molzan, Benjamin Schumacher, Corinna Ottmann, Angela Baljuls, Lisa Polzien, Michael Weyand, Philipp Thiel, Rolf Rose, Micheline Rose, Philipp Kuhenne, Markus Kaiser, Ulf R Rapp, Jürgen Kuhlmann, Christian Ottmann

Identification of novel in vivo phosphorylation sites of the human proapoptotic protein BAD: pore-forming activity of BAD is regulated by phosphorylation

鉴定人类促凋亡蛋白 BAD 的新型体内磷酸化位点:BAD 的成孔活性受磷酸化调控

Lisa Polzien, Angela Baljuls, Ulrike E E Rennefahrt, Andreas Fischer, Werner Schmitz, Rene P Zahedi, Albert Sickmann, Renate Metz, Stefan Albert, Roland Benz, Mirko Hekman, Ulf R Rapp