日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Molecular recognition at the opioid-modulating neuropeptide FF receptor 1

阿片类调节神经肽FF受体1的分子识别

Na, Man; Yue, Yang; Xu, Kexin; Xu, Ziyi; Zhang, Lu; Zhou, Fangfang; De Neve, Jolien; Ballet, Steven; Xu, Fei

Trifluoromethylthio and Trifluoromethyl Functionalization of Endomorphin-1 Enhances its Hydrophobicity and Plasma Stability while Preserving its Affinity for the μ-Opioid Receptor

内啡肽-1的三氟甲基硫代和三氟甲基功能化增强了其疏水性和血浆稳定性,同时保持了其对μ-阿片受体的亲和力。

Gregorc, Jure; De Neve, Jolien; Guitot, Karine; Holleran, Brian J; Lensen, Nathalie; Gendron, Louis; Brigaud, Thierry; Iskra, Jernej; Ballet, Steven; Chaume, Grégory

Developing nanobodies as allosteric molecular chaperones of glucocerebrosidase function.

开发纳米抗体作为葡糖脑苷脂酶功能的变构分子伴侣

Dal Maso Thomas, Sinisgalli Chiara, Zilio Gianluca, Franzin Elisa, Tessari Isabella, Pardon Els, Steyaert Jan, Ballet Steven, Greggio Elisa, Versées Wim, Plotegher Nicoletta

Inhibitors of Tax1-PDZ Interactions Block HTLV-1 Viral Transmission by Changing EV Composition.

Tax1-PDZ相互作用抑制剂通过改变EV组成阻断HTLV-1病毒传播

Puttemans Jedidja, Brammerloo Yasmine, Blibek Karim, Blavier Jeremy, Ntombela Thandokuhle, Van Molle Inge, Joseph Julie, Olivet Julien, Saha Deeya, Degey Manon, Hamaidia Malik, Jain Pooja, Geraldine Piel, Zimmermann Pascale, Kim Dae-Kyum, Baiwir Dominique, Njock Makon-Sébastien, Dequiedt Franck, Salehi-Ashtiani Kourosh, Ballet Steven, Volkov Alexander N, Twizere Jean-Claude, Maseko Sibusiso B

Peptide hydrogel-drug conjugates for tailored disease treatment

用于个体化疾病治疗的肽水凝胶-药物偶联物

Cauwenbergh, Thibault; Ballet, Steven; Martin, Charlotte

A short amphipathic peptide-based injectable hydrogel with antibacterial properties

一种具有抗菌性能的短链两亲性肽基可注射水凝胶

Aerssens, Dorien; Theppawong, Atiruj; Vu, Hue; Rigole, Petra; Van Troys, Marleen; Coenye, Tom; Hoogenboom, Richard; Ballet, Steven; Martin, Charlotte; Madder, Annemieke

Discovery and Characterization of a Selective Inhibitor of Synaptojanin1 5‑Phosphatase Activity

突触素1 5-磷酸酶活性选择性抑制剂的发现与表征

Martin, Ella; Giakoumakis, Danaë; Paesmans, Jone; Bisi, Nicolò; Drozdzecki, Andrzej; Audenaert, Dominique; Haustraete, Jurgen; Verstreken, Patrik; Galicia, Christian; Ballet, Steven; Versées, Wim

Design and synthesis of cyclic lipidated peptides derived from the C-terminus of Cx43 for hemichannel inhibition and cardiac endothelium targeting

设计和合成源自Cx43 C端环状脂化肽,用于半通道抑制和心脏内皮靶向治疗。

Iaculli, Debora; Montgomery, Jade; Lamouroux, Arthur; Caufriez, Anne; Gozalbes, Rafael; Vinken, Mathieu; Molica, Filippo; Kwak, Brenda R; Ballet, Steven

Allosteric nanobodies to study the interactions between SOS1 and RAS

利用变构纳米抗体研究SOS1与RAS之间的相互作用

Fischer, Baptiste; Uchański, Tomasz; Sheryazdanova, Aidana; Gonzalez, Simon; Volkov, Alexander N; Brosens, Elke; Zögg, Thomas; Kalichuk, Valentina; Ballet, Steven; Versées, Wim; Sablina, Anna A; Pardon, Els; Wohlkönig, Alexandre; Steyaert, Jan

Design, Synthesis, and In Vitro Characterization of Proteolytically-Stable Opioid-Neurotensin Hybrid Peptidomimetics

蛋白水解稳定的阿片-神经降压素杂合肽模拟物的设计、合成和体外表征

De Neve, Jolien; Breault, Émile; Previti, Santo; Vangeloven, Esaü; Loranger, Bobbi; Chartier, Magali; Brouillette, Rebecca; Lanoie, Annik; Holleran, Brian J; Longpré, Jean-Michel; Gendron, Louis; Tourwé, Dirk; Sarret, Philippe; Ballet, Steven