日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

ML314: A Biased Neurotensin Receptor Ligand for Methamphetamine Abuse

ML314:一种用于治疗甲基苯丙胺滥用的偏向性神经降压素受体配体

Barak, Larry S; Bai, Yushi; Peterson, Sean; Evron, Tama; Urs, Nikhil M; Peddibhotla, Satyamaheshwar; Hedrick, Michael P; Hershberger, Paul; Maloney, Patrick R; Chung, Thomas D Y; Rodriguiz, Ramona M; Wetsel, William C; Thomas, James B; Hanson, Glen R; Pinkerton, Anthony B; Caron, Marc G

Design, synthesis, and analysis of antagonists of GPR55: Piperidine-substituted 1,3,4-oxadiazol-2-ones

GPR55拮抗剂的设计、合成和分析:哌啶取代的1,3,4-恶二唑-2-酮

Meza-Aviña, Maria Elena; Lingerfelt, Mary A; Console-Bram, Linda M; Gamage, Thomas F; Sharir, Haleli; Gettys, Kristen E; Hurst, Dow P; Kotsikorou, Evangelia; Shore, Derek M; Caron, Marc G; Rao, Narasinga; Barak, Larry S; Abood, Mary E; Reggio, Patricia H; Croatt, Mitchell P

Perhexiline promotes HER3 ablation through receptor internalization and inhibits tumor growth.

哌克西林通过受体内化促进 HER3 消融,抑制肿瘤生长

Ren Xiu-Rong, Wang Jiangbo, Osada Takuya, Mook Robert A Jr, Morse Michael A, Barak Larry S, Lyerly Herbert Kim, Chen Wei

A rapid and affordable screening platform for membrane protein trafficking

一种快速且经济的膜蛋白转运筛选平台

Snyder, Joshua C; Pack, Thomas F; Rochelle, Lauren K; Chakraborty, Subhasish K; Zhang, Ming; Eaton, Andrew W; Bai, Yushi; Ernst, Lauren A; Barak, Larry S; Waggoner, Alan S; Caron, Marc G

The stem cell-expressed receptor Lgr5 possesses canonical and functionally active molecular determinants critical to β-arrestin-2 recruitment.

干细胞表达的受体 Lgr5 具有典型的、功能活跃的分子决定簇,对 β-arrestin-2 的募集至关重要

Snyder Joshua C, Rochelle Lauren K, Barak Larry S, Caron Marc G

Small molecule modulators of Wnt/β-catenin signaling

Wnt/β-catenin信号通路的小分子调节剂

Mook, Robert A Jr; Chen, Minyong; Lu, Jiuyi; Barak, Larry S; Lyerly, H Kim; Chen, Wei

BRET biosensors to study GPCR biology, pharmacology, and signal transduction

利用BRET生物传感器研究GPCR生物学、药理学和信号转导

Salahpour, Ali; Espinoza, Stefano; Masri, Bernard; Lam, Vincent; Barak, Larry S; Gainetdinov, Raul R

The insecticide synergist piperonyl butoxide inhibits hedgehog signaling: assessing chemical risks

杀虫剂增效剂胡椒基丁醚抑制 Hedgehog 信号通路:评估化学风险

Wang, Jiangbo; Lu, Jiuyi; Mook, Robert A Jr; Zhang, Min; Zhao, Shengli; Barak, Larry S; Freedman, Jonathan H; Lyerly, H Kim; Chen, Wei

Functional interaction between trace amine-associated receptor 1 and dopamine D2 receptor

痕量胺相关受体1与多巴胺D2受体之间的功能性相互作用

Espinoza, Stefano; Salahpour, Ali; Masri, Bernard; Sotnikova, Tatyana D; Messa, Mirko; Barak, Larry S; Caron, Marc G; Gainetdinov, Raul R

Glucocorticoid hedgehog agonists in neurogenesis

糖皮质激素和刺猬信号通路激动剂在神经发生中的作用

Wang, Jiangbo; Barak, Larry S; Mook, Robert A Jr; Chen, Wei