日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Population pharmacokinetic modelling of cetirizine concentrations in human breast milk-A contribution from the ConcePTION project

西替利嗪在人乳中的浓度群体药代动力学模型——来自 ConcePTION 项目的贡献

Melander, Erik; Nielsen, Elisabet I; Lindqvist, Annika; Hovd, Markus; Gandia, Peggy; Panchaud, Alice; Guidi, Monia; Annaert, Pieter; Baranczewski, Pawel; Spigset, Olav; Nordeng, Hedvig

AlphaFold accelerated discovery of psychotropic agonists targeting the trace amine-associated receptor 1

AlphaFold 加速发现针对微量胺相关受体 1 的精神药物激动剂

Alejandro Díaz-Holguín, Marcus Saarinen, Duc Duy Vo, Andrea Sturchio, Niclas Branzell, Israel Cabeza de Vaca, Huabin Hu, Núria Mitjavila-Domènech, Annika Lindqvist, Pawel Baranczewski, Mark J Millan, Yunting Yang, Jens Carlsson, Per Svenningsson

Antibiotic class with potent in vivo activity targeting lipopolysaccharide synthesis in Gram-negative bacteria

一类具有强效体内活性的抗生素,靶向革兰氏阴性菌脂多糖的合成。

Huseby, Douglas L; Cao, Sha; Zamaratski, Edouard; Sooriyaarachchi, Sanjeewani; Ahmad, Shabbir; Bergfors, Terese; Krasnova, Laura; Pelss, Juris; Ikaunieks, Martins; Loza, Einars; Katkevics, Martins; Bobileva, Olga; Cirule, Helena; Gukalova, Baiba; Grinberga, Solveiga; Backlund, Maria; Simoff, Ivailo; Leber, Anna T; Berruga-Fernández, Talía; Antonov, Dmitry; Konda, Vivekananda R; Lindström, Stefan; Olanders, Gustav; Brandt, Peter; Baranczewski, Pawel; Vingsbo Lundberg, Carina; Liepinsh, Edgars; Suna, Edgars; Jones, T Alwyn; Mowbray, Sherry L; Hughes, Diarmaid; Karlén, Anders

Targeted NUDT5 inhibitors block hormone signaling in breast cancer cells

靶向 NUDT5 抑制剂阻断乳腺癌细胞中的激素信号传导

Brent D G Page, Nicholas C K Valerie, Roni H G Wright, Olov Wallner, Rebecka Isaksson, Megan Carter, Sean G Rudd, Olga Loseva, Ann-Sofie Jemth, Ingrid Almlöf, Jofre Font-Mateu, Sabin Llona-Minguez, Pawel Baranczewski, Fredrik Jeppsson, Evert Homan, Helena Almqvist, Hanna Axelsson, Shruti Regmi, Anna

Anti-Rift Valley fever virus activity in vitro, pre-clinical pharmacokinetics and oral bioavailability of benzavir-2, a broad-acting antiviral compound

苯扎韦-2(一种广谱抗病毒化合物)的体外抗裂谷热病毒活性、临床前药代动力学和口服生物利用度

Islam, Md Koushikul; Strand, Mårten; Saleeb, Michael; Svensson, Richard; Baranczewski, Pawel; Artursson, Per; Wadell, Göran; Ahlm, Clas; Elofsson, Mikael; Evander, Magnus

Structure-metabolism-relationships in the microsomal clearance of piperazin-1-ylpyridazines

哌嗪-1-基哒嗪微粒体清除的结构-代谢关系

Llona-Minguez, Sabin; Ghassemian, Artin; Baranczewski, Pawel; Desroses, Matthieu; Koolmeister, Tobias; Artursson, Per; Scobie, Martin; Helleday, Thomas

Discovery of the First Potent and Selective Inhibitors of Human dCTP Pyrophosphatase 1

人类 dCTP 焦磷酸酶 1 的首个高效选择性抑制剂的发现

Llona-Minguez, Sabin; Höglund, Andreas; Jacques, Sylvain A; Johansson, Lars; Calderón-Montaño, José Manuel; Claesson, Magnus; Loseva, Olga; Valerie, Nicholas C K; Lundbäck, Thomas; Piedrafita, Javier; Maga, Giovanni; Crespan, Emmanuele; Meijer, Laurent; Morón, Estefanía Burgos; Baranczewski, Pawel; Hagbjörk, Ann-Louise; Svensson, Richard; Wiita, Elisee; Almlöf, Ingrid; Visnes, Torkild; Jeppsson, Fredrik; Sigmundsson, Kristmundur; Jensen, Annika Jenmalm; Artursson, Per; Jemth, Ann-Sofie; Stenmark, Pål; Berglund, Ulrika Warpman; Scobie, Martin; Helleday, Thomas