日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The Development of UM-203, A Reversible Covalent STING Antagonist

UM-203(一种可逆共价STING拮抗剂)的研制

Barasa, Leonard; DeOrsey, Leo; O'Reilly, Maeve D; Choudhary, Shruti; Cahill, Sara E; Mathur, Anukriti; Allabaji, Akumalla; Vidadala, Srinivasa Rao; Sarkar, Sujit Kumar; Patil, Santoshkumar N; Kalonia, Harikesh; Hale, Jeffrey; Humphries, Fiachra; Fitzgerald, Katherine A; Thompson, Paul R

Triazole-based STING inhibitors

基于三唑的STING抑制剂

Singh, Anju; Barasa, Leonard; DeOrsey, Leo; O'Reilly, Maeve D; Choudhary, Shruti; Cahill, Sara E; Rossetti, Thomas; Green, Robert Madison; Humphries, Fiachra; Thompson, Paul R

Reciprocal regulation between the protein arginine deiminases and mSWI/SNF chromatin remodelers controls skeletal muscle differentiation and regeneration

蛋白质精氨酸脱亚胺酶与mSWI/SNF染色质重塑因子之间的相互调控控制着骨骼肌的分化和再生。

Olea-Flores, Monserrat; Sharma, Tapan; Parikh, Anand; Barasa, Leonard; Hachmer, Sarah; Dilworth, F Jeffrey; Padilla-Benavides, Teresita; Thompson, Paul R; Imbalzano, Anthony N

Multifunctional Conductive Nanofibers for Self‐Powered Glucose Biosensors (Adv. Sci. 18/2025)

用于自供电葡萄糖生物传感器的多功能导电纳米纤维(Adv. Sci. 18/2025)

Yang, Shengjie; Xue, Jiaqi; Li, Ziqi; Zhang, Shiqing; Zhang, Zhang; Huang, Zhifeng; Yung, Ken Kin Lam; Lai, King Wai Chiu; Brennan, Andrew; Lovell, Scott; Vance, Keith W; Mason, Jody M; Yu, Xin; Song, Yujing; Dong, Tao; Ouyang, Wenlu; Quan, Chao; Shao, Liujiazi; Barasa, Leonard; Thompson, Paul R; Zhang, Mao; Ma, Jianjie; Kurabayashi, Katsuo; Li, Yongqing; Ou, Zhihua; Li, Li; Ren, Peidi; Zhou, Ting‐Ting; He, Fan; Chen, Jialing; Cai, Huimin; Han, Xiumin; Wu, Yao‐Dong; Li, Jiandong; Li, Xiu‐Rong; Tan, Qiming; Li, Wenhui; Chen, Qi; Zhang, Nian‐Zhang; He, Xiuju; Chen, Wei‐Gang; Zhao, Yanping; Sun, Jiwen; Zhang, Qian; Wu, Yan‐Tao; Liang, Yingan; You, Jie; Hu, Guohai; Tian, Xue‐Qi; Liao, Sha; Fu, Bao‐Quan; Chen, Ao; Cai, Xue‐Peng; Yang, Huanming; Wang, Jian; Jin, Xin; Xu, Xun; Jia, Wan‐Zhong; Li, Junhua; Yan, Hong‐Bin; Feng, Xiaodan; Xu, Xinran; Meng, Zhaonan; Jiang, Jiahao; Pei, Miao; Zheng, Yonghe; Lu, Chunming; Zhang, Guangyu; Zhang, Xin; Pan, Wenting; Chen, Xizhao; Wan, Lingfei; Liu, Chunjie; Yong, Yuting; Zhao, Yue; Sang, Shuli; Zhang, Lihua; Yao, Sheng; Guo, Yushu; Wang, Mingmei; Wang, Xinhui; Peng, Guangdun; Yan, Xinlong; Wang, Yanchun; Zhang, Min; Ciccone, Giuseppe; Azevedo Gonzalez‐Oliva, Mariana; Versaevel, Marie; Cantini, Marco; Vassalli, Massimo; Salmeron‐Sanchez, Manuel; Gabriele, Sylvain; Xu, Qingmei; Wang, Yuntong; Dou, Songtao; Xu, Yang; Xu, Zhenhe; Xu, Han; Zhang, Yi; Xia, Yanming; Xue, Ying; Li, Hang; Ma, Xiao; Zhang, Kunlong; Wang, Huan; Ma, Fengzhou; Wang, Qi; Li, Bei; Wang, Wei; Li, Haoran; Luo, Kang; Tsai, Din Ping; Li, Yulang; Dou, Linyuan; Li, Shuqiao; He, Tao; Fan, Yuancheng; Chen, Mu Ku; Wang, Zhanshan; Shi, Yuzhi; Wei, Zeyong; Cheng, Xinbin; Gungordu Er, Seda; Bulathsinghala, Rameesh; Kizilates, Selvinaz Burcu; Li, Bing; Ryan, Rucchi; Tabish, Tanveer A; Dharmasena, Ishara; Edirisinghe, Mohan

Citrullination of NF-κB p65 by PAD2 as a Novel Therapeutic Target for Modulating Macrophage Polarization in Acute Lung Injury.

PAD2介导的NF-κB p65瓜氨酸化是调节急性肺损伤中巨噬细胞极化的新型治疗靶点

Yu Xin, Song Yujing, Dong Tao, Ouyang Wenlu, Quan Chao, Shao Liujiazi, Barasa Leonard, Thompson Paul R, Zhang Mao, Ma Jianjie, Kurabayashi Katsuo, Li Yongqing

Nitrofuran-Based STING Inhibitors

基于硝基呋喃的STING抑制剂

Barasa, Leonard; DeOrsey, Leo; O'Reilly, Maeve D; Choudhary, Shruti; Cahill, Sara E; Mathur, Anukriti; Rajoria, Sakshi; Green, Robert Madison; Allabaji, Akumalla; Nellikkalaya, Shreekrishna; Paul, Sourav; Vidadala, Srinivasa Rao; Kumar Sarkar, Sujit; Patil, Santoshkumar N; Hale, Jeffrey; Humphries, Fiachra; Fitzgerald, Katherine A; Thompson, Paul R

N,N-Diethylacetamide and N,N-Dipropylacetamide inhibit the NF-kB pathway in in vitro, ex vivo and in vivo models of inflammation-induced preterm birth

N,N-二乙基乙酰胺和N,N-二丙基乙酰胺在体外、离体和体内炎症诱导早产模型中均能抑制NF-κB通路。

Gorasiya, Samir; Mushi, Juliet; Yoganathan, Sabesan; Barasa, Leonard; Pekson, Ryan; Ashby, Charles R Jr; Reznik, Sandra E

High-Throughput Screening of More Than 30,000 Compounds for Anthelmintics against Gastrointestinal Nematode Parasites.

对超过 30,000 种化合物进行高通量筛选,以寻找对抗胃肠道线虫寄生虫的驱虫药

Elfawal Mostafa A, Goetz Emily, Kim Youmie, Chen Paulina, Savinov Sergey N, Barasa Leonard, Thompson Paul R, Aroian Raffi V

Protein citrullination: inhibition, identification and insertion

蛋白质瓜氨酸化:抑制、鉴定和插入

Barasa, Leonard; Thompson, Paul R

SARM1, an Enzyme Involved in Axon Degeneration, Catalyzes Multiple Activities through a Ternary Complex Mechanism

SARM1是一种参与轴突退化的酶,它通过三元复合物机制催化多种活性。

Icso, Janneke D; Barasa, Leonard; Thompson, Paul R