日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Shared host genetic landscape of respiratory viral infection

呼吸道病毒感染的共同宿主遗传图谱

Soriaga, Leah B; Balce, Dale R; Bartha, Istvan; Park, Arnold; Wong, Emily; McAllaster, Michael; Mueller, Elizabeth A; Barauskas, Ona; Carabajal, Esteban; Kowalski, Beatriz; Lee, Sooyoung; Lo, Gary; Mahoney, Tara F; Metruccio, Matteo; Sahakyan, Anna; Somasundaram, Logeshwaran; Steinfeld, Tod; Wang, Lisha; Wedel, Laura; Yim, Samantha S; Yin, Li; Zhou, Jiayi; Newby, Zach; Tse, Winston; Grosse, Johannes; Virgin, Herbert W; Hwang, Seungmin; Telenti, Amalio

Discovery of Potent and Selective MTH1 Inhibitors for Oncology: Enabling Rapid Target (In)Validation

发现用于肿瘤治疗的高效选择性MTH1抑制剂:实现靶点(不)验证的快速开展

Farand, Julie; Kropf, Jeffrey E; Blomgren, Peter; Xu, Jianjun; Schmitt, Aaron C; Newby, Zachary E; Wang, Ting; Murakami, Eisuke; Barauskas, Ona; Sudhamsu, Jawahar; Feng, Joy Y; Niedziela-Majka, Anita; Schultz, Brian E; Schwartz, Karen; Viatchenko-Karpinski, Serge; Kornyeyev, Dmytro; Kashishian, Adam; Fan, Peidong; Chen, Xiaowu; Lansdon, Eric B; Ports, Michael O; Currie, Kevin S; Watkins, William J; Notte, Gregory T

Biochemical characterization of recombinant influenza A polymerase heterotrimer complex: Polymerase activity and mechanisms of action of nucleotide analogs

重组甲型流感病毒聚合酶异源三聚体复合物的生化特性:聚合酶活性和核苷酸类似物的作用机制

Barauskas, Ona; Xing, Weimei; Aguayo, Esmeralda; Willkom, Madeleine; Sapre, Annapurna; Clarke, Michael; Birkus, Gabriel; Schultz, Brian E; Sakowicz, Roman; Kwon, HyockJoo; Feng, Joy Y

Biochemical characterization of recombinant influenza A polymerase heterotrimer complex: Endonuclease activity and evaluation of inhibitors.

重组甲型流感聚合酶异三聚体复合物的生化特性:核酸内切酶活性及抑制剂评价

Xing Weimei, Barauskas Ona, Kirschberg Thorsten, Niedziela-Majka Anita, Clarke Michael, Birkus Gabriel, Weissburg Perry, Liu Xiaohong, Schultz Brian E, Sakowicz Roman, Kwon HyockJoo, Feng Joy Y

Structural and regulatory elements of HCV NS5B polymerase--β-loop and C-terminal tail--are required for activity of allosteric thumb site II inhibitors

HCV NS5B聚合酶的结构和调控元件——β环和C端尾部——是变构拇指位点II抑制剂发挥活性所必需的。

Boyce, Sarah E; Tirunagari, Neeraj; Niedziela-Majka, Anita; Perry, Jason; Wong, Melanie; Kan, Elaine; Lagpacan, Leanna; Barauskas, Ona; Hung, Magdeleine; Fenaux, Martijn; Appleby, Todd; Watkins, William J; Schmitz, Uli; Sakowicz, Roman

Secretory leukocyte protease inhibitor binds to Neisseria gonorrhoeae outer membrane opacity protein and is bactericidal

分泌型白细胞蛋白酶抑制剂与淋病奈瑟菌外膜不透明蛋白结合,具有杀菌作用。

Cooper, Morris D; Roberts, Melissa H; Barauskas, Ona L; Jarvis, Gary A