日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Rapidly expanded partially HLA DRB1-matched fungus-specific T cells mediate in vitro and in vivo antifungal activity

快速扩增的部分HLA-DRB1匹配的真菌特异性T细胞介导体外和体内抗真菌活性

Castellano-González, Gloria; McGuire, Helen M; Luciani, Fabio; Clancy, Leighton E; Li, Ziduo; Avdic, Selmir; Hughes, Brendan; Singh, Mandeep; Fazekas de St Groth, Barbara; Renga, Giorgia; Pariano, Marilena; Bellet, Marina M; Romani, Luigina; Gottlieb, David J

Navigation in bile acid chemical space: discovery of novel FXR and GPBAR1 ligands

胆汁酸化学空间导航:发现新型 FXR 和 GPBAR1 配体

Claudia Finamore, Carmen Festa, Barbara Renga, Valentina Sepe, Adriana Carino, Dario Masullo, Michele Biagioli, Silvia Marchianò, Angela Capolupo, Maria Chiara Monti, Stefano Fiorucci, Angela Zampella

Insights on FXR selective modulation. Speculation on bile acid chemical space in the discovery of potent and selective agonists

对 FXR 选择性调节的见解。对胆汁酸化学空间在发现强效和选择性激动剂中的推测

Valentina Sepe, Carmen Festa, Barbara Renga, Adriana Carino, Sabrina Cipriani, Claudia Finamore, Dario Masullo, Federica Del Gaudio, Maria Chiara Monti, Stefano Fiorucci, Angela Zampella

Structure-based drug design targeting the cell membrane receptor GPBAR1: exploiting the bile acid scaffold towards selective agonism

针对细胞膜受体 GPBAR1 的基于结构的药物设计:利用胆汁酸支架实现选择性激动

Francesco Saverio Di Leva, Carmen Festa, Barbara Renga, Valentina Sepe, Ettore Novellino, Stefano Fiorucci, Angela Zampella, Vittorio Limongelli

The HIV matrix protein p17 induces hepatic lipid accumulation via modulation of nuclear receptor transcriptoma

HIV 基质蛋白 p17 通过调节核受体转录瘤诱导肝脏脂质积累

Barbara Renga, Daniela Francisci, Adriana Carino, Silvia Marchianò, Sabrina Cipriani, Maria Chiara Monti, Rachele Del Sordo, Elisabetta Schiaroli, Eleonora Distrutti, Franco Baldelli, Stefano Fiorucci

Impaired Itching Perception in Murine Models of Cholestasis Is Supported by Dysregulation of GPBAR1 Signaling

胆汁淤积小鼠模型中的瘙痒感知受损是由 GPBAR1 信号失调引起的

Sabrina Cipriani, Barbara Renga, Claudio D'Amore, Michele Simonetti, Antonio Angelo De Tursi, Adriana Carino, Maria Chiara Monti, Valentina Sepe, Angela Zampella, Stefano Fiorucci

Marine and semi-synthetic hydroxysteroids as new scaffolds for pregnane X receptor modulation

海洋和半合成羟基类固醇作为孕烷 X 受体调节的新支架

Valentina Sepe, Francesco Saverio Di Leva, Claudio D'Amore, Carmen Festa, Simona De Marino, Barbara Renga, Maria Valeria D'Auria, Ettore Novellino, Vittorio Limongelli, Lisette D'Souza, Mahesh Majik, Angela Zampella, Stefano Fiorucci

The HIV matrix protein p17 promotes the activation of human hepatic stellate cells through interactions with CXCR2 and Syndecan-2

HIV 基质蛋白 p17 通过与 CXCR2 和 Syndecan-2 相互作用促进人类肝星状细胞的活化

Barbara Renga, Daniela Francisci, Elisabetta Schiaroli, Adriana Carino, Sabrina Cipriani, Claudio D'Amore, Angelo Sidoni, Rachele Del Sordo, Ivana Ferri, Monica Lucattelli, Benedetta Lunghi, Franco Baldelli, Stefano Fiorucci

Activation of the bile acid receptor GPBAR1 protects against gastrointestinal injury caused by non-steroidal anti-inflammatory drugs and aspirin in mice

激活胆汁酸受体 GPBAR1 可保护小鼠免受非甾体抗炎药和阿司匹林引起的胃肠道损伤

Sabrina Cipriani, Andrea Mencarelli, Angela Bruno, Barbara Renga, Eleonora Distrutti, Luca Santucci, Franco Baldelli, Stefano Fiorucci

Solomonsterol A, a marine pregnane-X-receptor agonist, attenuates inflammation and immune dysfunction in a mouse model of arthritis

Solomonsterol A 是一种海洋孕烷-X 受体激动剂,可减轻小鼠关节炎模型中的炎症和免疫功能障碍

Andrea Mencarelli, Claudio D'Amore, Barbara Renga, Sabrina Cipriani, Adriana Carino, Valentina Sepe, Elisa Perissutti, Maria Valeria D'Auria, Angela Zampella, Eleonora Distrutti, Stefano Fiorucci