日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

First-in-class SAM-competitive G9a inhibitor FLAV-27 as a disease-modifying therapy for Alzheimer disease.

首个SAM竞争性G9a抑制剂FLAV-27作为阿尔茨海默病疾病修饰疗法。

Bellver-Sanchis Aina, Valle-Garcia David, Barbaraci Carla, Romero-Becerra Fernando, Singh Rohit Kumar, Jarne-Ferrer Júlia, Vasilopoulou Foteini, Irisarri Alba, Martínez-Fernández Carmen, Fafián-Labora Juan A, Arufe María C, Wüst Carolin, Castellanos Aida, Soto David, Casals Núria, Fadó Rut, Pocock Jennifer M, Navarro Gemma, Val Cristina, Brea José, Loza M Isabel, Lleó Albert, Fortea Juan, Alcolea Daniel, Perez-Bosque Anna, Miró Lluïsa, Pérez Belén, Rashid Sajid, Ali Muhammad, Saqib Manahil, Lí Carbó Marcel, Guerrero Ana, Vázquez Santiago, Choudhary Bhanwar Singh, Dai Shaodong, Escolano Carmen, Franco Rafael, Pallàs Mercè, Griñán-Ferré Christian

Modulation of Tau Protein Neurotoxic Hallmarks by Novel σ(1)R Agonists/HDAC Inhibitor Dual-Acting Compounds

新型σ(1)R激动剂/HDAC抑制剂双效化合物对Tau蛋白神经毒性特征的调节

Fallica, Antonino N; Barbaraci, Carla; Ruiz-Cantero, M Carmen; Scarlatti, Arianna; Coco, Alessandro; Giordano, Giorgia; La Mantia, Alfonsina; Prezzavento, Orazio; Di Stefano, Antonio; Cacciatore, Ivana; Siano, Giacomo; Cattaneo, Antonino; Pasquinucci, Lorella; Cobos, Enrique J; Di Primio, Cristina; Amata, Emanuele; Marrazzo, Agostino

A brain-penetrant P2X7R antagonist mitigates Alzheimer's disease pathology

一种能穿透血脑屏障的P2X7R拮抗剂可减轻阿尔茨海默病病理。

Turcu, Andreea L; Oken, Adam C; Griñán-Ferré, Christian; Durner, Anna; Sierra-Marquez, Juan; Hinz-Kowalik, Sonja; Nagel, Jessica; Lee, So-Deok; Tzortzini, Efpraxia; Georgiou, Kyriakos; Bhol, Mamina; Baz, Zuriñe; Llop, Jordi; Schneider, Marion; Barbaraci, Carla; Kim, Ga-Ram; Barniol-Xicota, Marta; Val, Cristina; Brea, José; Loza, M Isabel; Pérez, Belén; Naesens, Lieve; Kolocouris, Antonios; Kim, Yong-Chul; Müller, Christa E; Nicke, Annette; Pallàs, Mercè; Mansoor, Steven E; Vázquez, Santiago

HDAC/σ1R Dual-Ligand as a Targeted Melanoma Therapeutic

HDAC/σ1R双配体作为靶向黑色素瘤治疗药物

Leotta, Claudia Giovanna; Barbaraci, Carla; Fiorito, Jole; Coco, Alessandro; di Giacomo, Viviana; Amata, Emanuele; Marrazzo, Agostino; Pitari, Giovanni Mario

Identification of Hyperelastic Material Parameters of Elastomers by Reverse Engineering Approach

利用逆向工程方法识别弹性体的超弹性材料参数

Yenigun, Burak; Gkouti, Elli; Barbaraci, Gabriele; Czekanski, Aleksander