日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of a Pseudomonas aeruginosa-specific small molecule targeting outer membrane protein OprH-LPS interaction by a multiplexed screen.

通过多重筛选发现了一种靶向铜绿假单胞菌外膜蛋白 OprH-LPS 相互作用的小分子

Poulsen Bradley E, Warrier Thulasi, Barkho Sulyman, Bagnall Josephine, Romano Keith P, White Tiantian, Yu Xiao, Kawate Tomohiko, Nguyen Phuong H, Raines Kyra, Ferrara Kristina, Golas A Lorelei, FitzGerald Michael, Boeszoermenyi Andras, Kaushik Virendar, Serrano-Wu Michael, Shoresh Noam, Hung Deborah T

High-Throughput Screening Tool to Identify Small Molecule Inhibitors of Telomerase

用于鉴定端粒酶小分子抑制剂的高通量筛选工具

Aquilanti, Elisa; Barkho, Sulyman; Bozinov, Vincent; Kageler, Lauren; Garrity-Janger, Max; Mesleh, Michael F; Horner, Steven; Ranaghan, Matthew J; Meyerson, Matthew

Structure and inhibition mechanisms of Mycobacterium tuberculosis essential transporter efflux protein A.

结核分枝杆菌必需转运蛋白外排蛋白A的结构和抑制机制。

Khandelwal Nitesh Kumar, Gupta Meghna, Gomez James E, Barkho Sulyman, Guan Ziqiang, Eng Ashley Y, Kawate Tomo, Balasubramani Sree Ganesh, Sali Andrej, Hung Deborah T, Stroud Robert M

An Iterative Approach Guides Discovery of the FabI Inhibitor Fabimycin, a Late-Stage Antibiotic Candidate with In Vivo Efficacy against Drug-Resistant Gram-Negative Infections

迭代方法指导FabI抑制剂法比霉素的发现,法比霉素是一种后期抗生素候选药物,对耐药革兰氏阴性菌感染具有体内疗效。

Parker, Erica N; Cain, Brett N; Hajian, Behnoush; Ulrich, Rebecca J; Geddes, Emily J; Barkho, Sulyman; Lee, Hyang Yeon; Williams, John D; Raynor, Malik; Caridha, Diana; Zaino, Angela; Shekhar, Mrinal; Muñoz, Kristen A; Rzasa, Kara M; Temple, Emily R; Hunt, Diana; Jin, Xiannu; Vuong, Chau; Pannone, Kristina; Kelly, Aya M; Mulligan, Michael P; Lee, Katie K; Lau, Gee W; Hung, Deborah T; Hergenrother, Paul J

Correction to "An Iterative Approach Guides Discovery of the FabI Inhibitor Fabimycin, a Late-Stage Antibiotic Candidate with In Vivo Efficacy against Drug-Resistant Gram-Negative Infections"

对“迭代方法指导发现FabI抑制剂法比霉素,一种对耐药革兰氏阴性菌感染具有体内疗效的后期抗生素候选药物”一文的更正

Parker, Erica N; Cain, Brett N; Hajian, Behnoush; Ulrich, Rebecca J; Geddes, Emily J; Barkho, Sulyman; Lee, Hyang Yeon; Williams, John D; Raynor, Malik; Caridha, Diana; Zaino, Angela; Rohde, Jason M; Zak, Mark; Shekhar, Mrinal; Muñoz, Kristen A; Rzasa, Kara M; Temple, Emily R; Hunt, Diana; Jin, Xiannu; Vuong, Chau; Pannone, Kristina; Kelly, Aya M; Mulligan, Michael P; Lee, Katie K; Lau, Gee W; Hung, Deborah T; Hergenrother, Paul J

Structural characterisation of the catalytic domain of botulinum neurotoxin X - high activity and unique substrate specificity

肉毒杆菌神经毒素X催化结构域的结构表征——高活性和独特的底物特异性

Masuyer, Geoffrey; Zhang, Sicai; Barkho, Sulyman; Shen, Yi; Henriksson, Linda; Košenina, Sara; Dong, Min; Stenmark, Pål

Allosteric switching of agonist/antagonist activity by a single point mutation in the interluekin-1 receptor antagonist, IL-1Ra

白细胞介素-1受体拮抗剂IL-1Ra的单点突变可导致激动剂/拮抗剂活性发生变构转换。

Hailey, Kendra L; Capraro, Dominique T; Barkho, Sulyman; Jennings, Patricia A