日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A synergistic interaction between PRMT5 and LSD1 inhibitors in AML.

PRMT5 和 LSD1 抑制剂在急性髓系白血病中存在协同作用。

Param Nesteene Joy, Arceci Elisa, Fiorentino Francesco, Pignata Luca, Torre Denis, Gutiérrez-Trejo Nayeli, Fong Jia Yi, Goy Pierre-Alexis, Han Brenda Y, Lambona Chiara, Di Bello Elisabetta, Castiello Carola, Barone Marco, Schwarz Megan, Arrowsmith Cheryl, Ito Koichi, Scherle Peggy, Wee Dave Keng Boon, Ndoye Steven, Tabaglio Tommaso, Jeyasekharan Anand D, Lakshmanan Manikandan, Cirilli Roberto, Habisch Hansjörg, Madl Tobias, Mattevi Andrea, Valente Sergio, Mai Antonello, Guccione Ernesto

Covalent adduct Grob fragmentation underlies LSD1 demethylase-specific inhibitor mechanism of action and resistance.

共价加合物 Grob 断裂是 LSD1 去甲基酶特异性抑制剂作用机制和耐药性的基础

Waterbury Amanda L, Caroli Jonatan, Zhang Olivia, Tuttle Paloma R, Liu Chao, Li Jiaming, Park Ji Sung, Hoenig Samuel M, Barone Marco, Furui Airi, Mattevi Andrea, Liau Brian B

Modulating the Binding Kinetics of Bruton's Tyrosine Kinase Inhibitors through Transition-State Effects

通过过渡态效应调节布鲁顿酪氨酸激酶抑制剂的结合动力学

Bravo, Eduardo Jr; Li, Yong; Lin, David Yin-Wei; Srinivasan, Bharath; Barone, Marco; Li, Stan Xiaogang; DelloRusso, Francesca; Rahiyanath, Anza Suneer; Corrionero, Ana; Alfonso, Patricia; Prendiville, Niall; Kozakov, Dima; Andreotti, Amy H; Tonge, Peter J

Uncoupling histone modification crosstalk by engineering lysine demethylase LSD1.

通过改造赖氨酸去甲基酶 LSD1 来解耦组蛋白修饰串扰

Lee Kwangwoon, Barone Marco, Waterbury Amanda L, Jiang Hanjie, Nam Eunju, DuBois-Coyne Sarah E, Whedon Samuel D, Wang Zhipeng A, Caroli Jonatan, Neal Katherine, Ibeabuchi Brian, Dhoondia Zuzer, Kuroda Mitzi I, Liau Brian B, Beck Samuel, Mattevi Andrea, Cole Philip A

Exploring attentional mechanisms underlying the gender homophily in equity crowdfunding decisions using web-based eye-tracking

利用基于网络的眼动追踪技术探索股权众筹决策中性别同质性背后的注意力机制

Barone, Marco; Bussoli, Candida; Fattobene, Lucrezia; Ling, Aiqing

Light-Driven Enzyme Catalysis: Ultrafast Mechanisms and Biochemical Implications

光驱动酶催化:超快机制及其生物化学意义

He, YongLe; Barone, Marco; Meech, Stephen R; Lukacs, Andras; Tonge, Peter J

Evolution, structure, and drug-metabolizing activity of mammalian prenylcysteine oxidases

哺乳动物异戊二烯基半胱氨酸氧化酶的进化、结构和药物代谢活性

Barone, Marco; Pizzorni, Letizia; Fraaije, Marco W; Mascotti, Maria L; Mattevi, Andrea

Asymmetric Engagement of Dimeric CRL3 (KBTBD4) by the Molecular Glue UM171 Licenses Degradation of HDAC1/2 Complexes

分子胶UM171与二聚体CRL3(KBTBD4)的不对称结合促进HDAC1/2复合物的降解

Yeo, Megan Jr; Zhang, Olivia; Xie, Xiaowen; Nam, Eunju; Payne, Neil Connor; Gosavi, Pallavi M; Kwok, Hui Si; Iram, Irtiza; Lee, Ceejay; Li, Jiaming; Chen, Nicholas J; Jiang, Hanjie; Wang, Zhipeng A; Lee, Kwangwoon; Mao, Haibin; Harry, Stefan A; Barakat, Idris A; Takahashi, Mariko; Waterbury, Amanda L; Barone, Marco; Mattevi, Andrea; Bar-Peled, Liron; Cole, Philip A; Mazitschek, Ralph; Liau, Brian B; Zheng, Ning

Computationally driven discovery of SARS-CoV-2 M(pro) inhibitors: from design to experimental validation

基于计算的SARS-CoV-2 M(pro)抑制剂发现:从设计到实验验证

El Khoury, Léa; Jing, Zhifeng; Cuzzolin, Alberto; Deplano, Alessandro; Loco, Daniele; Sattarov, Boris; Hédin, Florent; Wendeborn, Sebastian; Ho, Chris; El Ahdab, Dina; Jaffrelot Inizan, Theo; Sturlese, Mattia; Sosic, Alice; Volpiana, Martina; Lugato, Angela; Barone, Marco; Gatto, Barbara; Macchia, Maria Ludovica; Bellanda, Massimo; Battistutta, Roberto; Salata, Cristiano; Kondratov, Ivan; Iminov, Rustam; Khairulin, Andrii; Mykhalonok, Yaroslav; Pochepko, Anton; Chashka-Ratushnyi, Volodymyr; Kos, Iaroslava; Moro, Stefano; Montes, Matthieu; Ren, Pengyu; Ponder, Jay W; Lagardère, Louis; Piquemal, Jean-Philip; Sabbadin, Davide

The antidepressant fluoxetine acts on energy balance and leptin sensitivity via BDNF

抗抑郁药氟西汀通过 BDNF 作用于能量平衡和瘦素敏感性

Gaia Scabia, Ilaria Barone, Marco Mainardi, Giovanni Ceccarini, Manuela Scali, Emma Buzzigoli, Alessia Dattilo, Paolo Vitti, Amalia Gastaldelli, Ferruccio Santini, Tommaso Pizzorusso, Lamberto Maffei, Margherita Maffei