日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Characterization of PROTAC specificity and endogenous protein interactomes using ProtacID.

利用ProtacID对PROTAC特异性和内源性蛋白质相互作用组进行表征

Shrestha Suman, Maitland Matthew E R, Jing Laili, Duan Shili, Nie David Y, St-Germain Jonathan, Kanaris Michael, Barsyte-Lovejoy Dalia, Arrowsmith Cheryl H, Raught Brian

PRMT5 promotes full-length HTT expression by repressing multiple proximal intronic polyadenylation sites.

PRMT5 通过抑制多个近端内含子多聚腺苷酸化位点来促进全长 HTT 表达

Yadav Manisha, AlQazzaz Mona A, Ciamponi Felipe E, Ho Jolene C, Maron Maxim I, Sababi Aiden M, MacLeod Graham, Ahmadi Moloud, Bullivant Garrett, Tano Vincent, Langley Sarah R, Sánchez-Osuna María, Sachamitr Patty, Kushida Michelle, Bardile Costanza Ferrari, Pouladi Mahmoud A, Kurtz Rebecca, Richards Laura, Pugh Trevor, Tyers Mike, Angers Stephane, Dirks Peter B, Bader Gary D, Truant Ray, Massirer Katlin B, Barsyte-Lovejoy Dalia, Shechter David, Harding Rachel J, Arrowsmith Cheryl H, Prinos Panagiotis

PRMT1 inhibitor MS023 suppresses RNA splicing to sensitize small cell lung cancer to DNA damaging agents.

PRMT1 抑制剂 MS023 抑制 RNA 剪接,使小细胞肺癌对 DNA 损伤剂更加敏感

Aparnathi Mansi K, Ul Haq Sami, St-Germain Jonathan, Nixon Kevin C J, Walton Joseph, Song Lifang, Majeed Safa, Patel Parasvi S, Subramaniam Ratheesh, Philip Vivek, Marcellus Richard, Barsyte-Lovejoy Dalia, Al-Awar Rima, Hakem Razqallah, Arrowsmith Cheryl H, Ailles Laurie, Raught Brian, Lok Benjamin H

A Target Class Ligandability Evaluation of WD40 Repeat-Containing Proteins

WD40重复序列蛋白的靶向配体结合能力评价

Ackloo, Suzanne; Li, Fengling; Szewczyk, Magda; Seitova, Almagul; Loppnau, Peter; Zeng, Hong; Xu, Jin; Ahmad, Shabbir; Arnautova, Yelena A; Baghaie, A J; Beldar, Serap; Bolotokova, Albina; Centrella, Paolo A; Chau, Irene; Clark, Matthew A; Cuozzo, John W; Dehghani-Tafti, Saba; Disch, Jeremy S; Dong, Aiping; Dumas, Antoine; Feng, Jianwen A; Ghiabi, Pegah; Gibson, Elisa; Gilmer, Justin; Goldman, Brian; Green, Stuart R; Guié, Marie-Aude; Guilinger, John P; Harms, Nathan; Herasymenko, Oleksandra; Houliston, Scott; Hutchinson, Ashley; Kearnes, Steven; Keefe, Anthony D; Kimani, Serah W; Kramer, Trevor; Kutera, Maria; Kwak, Haejin A; Lento, Cristina; Li, Yanjun; Liu, Jenny; Loup, Joachim; Machado, Raquel A C; Mulhern, Christopher J; Perveen, Sumera; Righetto, Germanna L; Riley, Patrick; Shrestha, Suman; Sigel, Eric A; Silva, Madhushika; Sintchak, Michael D; Slakman, Belinda L; Taylor, Rhys D; Thompson, James; Torng, Wen; Underkoffler, Carl; von Rechenberg, Moritz; Walsh, Ryan T; Watson, Ian; Wilson, Derek J; Wolf, Esther; Yadav, Manisha; Yazdi, Aliakbar K; Zhang, Junyi; Zhang, Ying; Santhakumar, Vijayaratnam; Edwards, Aled M; Barsyte-Lovejoy, Dalia; Schapira, Matthieu; Brown, Peter J; Halabelian, Levon; Arrowsmith, Cheryl H

OICR-41103 as a chemical probe for the DCAF1 WD40 domain.

OICR-41103 作为 DCAF1 WD40 结构域的化学探针

Kimani Serah W, Noureldin Mahmoud, Wilson Brian, Hoffer Laurent, Green Stuart R, Szewczyk Magdalena M, González-Álvarez Héctor, Mohammed Mohammed, Chan Manuel, Krausser Chiara, Li Alice Shi Ming, Hajian Taraneh, Tucker Sarah, Joshi Dhananjay, Saraon Punit, Thériault Brigitte, Kim Ji Sup, Santhakumar Vijayaratnam, Loppnau Peter, Li Yanjun, Seitova Almagul, Dong Aiping, Kiyota Taira, Hammann Tobias, Gehrtz Paul, Patel Bhashant, Rathod Vaibhavi, Vala Anand, Rout Bhimsen, Jagodra Paras, Brown Peter J, Aman Ahmed, Ramnauth Jailall, Poda Gennady, Uehling David, Arrowsmith Cheryl H, Barsyte-Lovejoy Dalia, Marcellus Richard, Ackloo Suzanne, Mamai Ahmed, Al-Awar Rima, Halabelian Levon

Musculoskeletal Disorders among Lithuanian Dentists and Oral Hygienists

立陶宛牙医和口腔卫生员的肌肉骨骼疾病

Barsyte, Eigile; Bineviciute, Zemyna; Venskutonis, Tadas

Everyday norms have become more permissive over time and vary across cultures

随着时间的推移,日常规范变得更加宽松,并且因文化而异。

Eriksson, Kimmo; Strimling, Pontus; Vartanova, Irina; Simpson, Brent; Persson, Minna; Abdi, Khalid Ahmed; Ad, Neta; Aldashev, Alisher; Ali, Habib Mohammad; Alì, Maurizio; Aliyev, Khatai; Alrefaee, Yasser M H A; Alvarado Ortiz, Alberth Estuardo; Andersson, Per A; Andrighetto, Giulia; Arikan, Gizem; Aruta, John Jamir Benzon R; Ayikwa, Christian Lutete; Baños-Chaparro, Jonatan; Barrera, Davide; Barsyte, Justina; Batkeyev, Birzhan; Batool, Azma; Berezina, Elizaveta; Bimina, Stéphanie Ngandu; Björnstjerna, Marie; Blumen, Sheyla; Boski, Paweł; Boštjančič, Eva; Boum, Yap 2nd; Briguglio, Marie; Bruno, Kagonbe; Bui, Huyen Thi Thu; Caycho-Rodríguez, Tomás; Chen, Yanyan; Chiweshe, Manase Kudzai; Choi, Hoon-Seok; Contreras-Ibáñez, Carlos C; Čorkalo, Dinka; Cruz-Torres, Christian E; Czakó, Andrea; de Zoysa, Piyanjali; Demetrovics, Zsolt; Dinić, Bojana M; Drače, Saša; El-Haddad, Rita W; Engelmann, Jan B; Escudero Pérez, Ignacio; Euh, Hyun; Fang, Xia; Frank, Celine; Freidin, Esteban; Fulop, Marta; Gamsakhurdia, Vladimer; García Jiménez, Mauro Alberto; Gardarsdottir, Ragna B; Gavreliuc, Alin; Gill, Colin Mathew Hugues D; Gjoneska, Biljana; Glöckner, Andreas; Graf, Sylvie; Grigoryan, Ani; Growiec, Katarzyna; Haas, Brian W; Haddock, Geoffrey; Hadjisolomou, Stavros P; Hadžiahmetović, Nina; Haji Mohammad Ali, Mohammad Hosein; Hakoköngäs, Eemeli; Halama, Peter; Hapunda, Given; Hartanto, Andree; Hazrati, Mahsa; Herbas-Torrico, Boris Christian; Holka, Szilárd; Hřebíčková, Martina; Hunter, John A; Ibikounle, Moudachirou; Ilisko, Dzintra; Lind Hjördísar Jónsdóttir, Harpa; Kaminskiene, Zivile; Kapoor, Hansika; Kapović, Iva; Karim, Gassemi; Kawakami, Kerry; Khachatryan, Narine; Kirschner, Julian B; Kiruja, Jonah; Kiyonari, Toko; Kohút, Michal; Kousar, Shazia; Krasniqi, Besnik; Lado, Ludovic; Landa-Blanco, Miguel; Landon, Barbara; Lep, Žan; Leslie, Lisa M; Li, Yang; Liik, Kadi; Lin, Ming-Jen; Lobos Rivera, Marlon Elías; López-López, Wilson; Maloku, Edona; Mandal, Mohona; Manhique, Bernardo Ananias; Mbende, Nathan Mpeti; Medhioub, Imed; Teixeira, Maria Luisa Mendes; Merchán Tamayo, J Paola; Mohammed, Linda Lila; Moore, Schontal N; Moraligil, Bahar; Muradzada, Nijat; Nanda, Herwin; Nastina, Ekaterina; Nejat, Pegah; Nettle, Daniel; Nipassa, Orlando Julio Andre; Noe-Grijalva, Martin; Ntampaka, Pie; Ntone, Rodrigue; Nussinson, Ravit; Oljača, Milan; Onyedire, Nneoma G; Onyishi, Ike E; Panagiotopoulou, Penny; Alvarez, Daybel Pañellas; Parvez, Md Shahin; Pasin, Gian Luca; Pedović, Ivana; Pérez de León, Pablo; Perez Floriano, Lorena R; Pop-Jordanova, Nada; Portillo, Jose Roberto; Potang, Angela; Quesada-Román, Adolfo; Raver, Jana L; Rodrigues, Ricardo B; Rodríguez-Romero, Juan Diego; Romanò, Sara; Ross, Robert M; Rosun, Nachita; Sadiković, Selka; San Martin, Alvaro; Smederevac, Snežana; Smith, Sarah Jane; Soboleva, Natalia; Sonessa, Daniel Erena; Stanley, Samantha K; Stoyanova, Kristina; Stoyanov, Drozdstoy; Takemura, Kosuke; Thøgersen, John; Tiliouine, Habib; Tung, Hans; Ulambayar, Tungalag; Uzdavinyte, Elze Marija; Waechter, Randall; Wang, Yi-Ting; Wu, Junhui; Yambio, Brice Martial; Yankson, Eric; Yeh, Kuang-Hui; Van Lange, Paul A M

Crystal structures of DCAF1-PROTAC-WDR5 ternary complexes provide insight into DCAF1 substrate specificity

DCAF1-PROTAC-WDR5三元复合物的晶体结构揭示了DCAF1的底物特异性

Mark F Mabanglo # ,Brian Wilson # ,Mahmoud Noureldin # ,Serah W Kimani ,Ahmed Mamai ,Chiara Krausser ,Héctor González-Álvarez ,Smriti Srivastava ,Mohammed Mohammed ,Laurent Hoffer ,Manuel Chan ,Jamie Avrumutsoae ,Alice Shi Ming Li ,Taraneh Hajian ,Sarah Tucker ,Stuart Green ,Magdalena Szewczyk ,Dalia Barsyte-Lovejoy ,Vijayaratnam Santhakumar ,Suzanne Ackloo ,Peter Loppnau ,Yanjun Li ,Almagul Seitova ,Taira Kiyota ,Jue George Wang ,Gilbert G Privé ,Douglas A Kuntz ,Bhashant Patel ,Vaibhavi Rathod ,Anand Vala ,Bhimsen Rout ,Ahmed Aman ,Gennady Poda ,David Uehling ,Jailall Ramnauth ,Levon Halabelian ,Richard Marcellus ,Rima Al-Awar ,Masoud Vedadi

Loss-of-function mutation in PRMT9 causes abnormal synapse development by dysregulation of RNA alternative splicing

PRMT9 的功能丧失突变通过 RNA 可变剪接失调导致突触发育异常

Lei Shen #, Xiaokuang Ma #, Yuanyuan Wang #, Zhihao Wang, Yi Zhang, Hoang Quoc Hai Pham, Xiaoqun Tao, Yuehua Cui, Jing Wei, Dimitri Lin, Tharindumala Abeywanada, Swanand Hardikar, Levon Halabelian, Noah Smith, Taiping Chen, Dalia Barsyte-Lovejoy, Shenfeng Qiu, Yi Xing, Yanzhong Yang

Recruitment of FBXO22 for targeted degradation of NSD2

FBXO22 的募集用于靶向降解 NSD2

David Y Nie #,John R Tabor #,Jianping Li,Maria Kutera,Jonathan St-Germain,Ronan P Hanley,Esther Wolf,Ethan Paulakonis,Tristan M G Kenney,Shili Duan,Suman Shrestha,Dominic D G Owens,Matthew E R Maitland,Ailing Pon,Magdalena Szewczyk,Anthony Joseph Lamberto,Michael Menes,Fengling Li,Linda Z Penn,Dalia Barsyte-Lovejoy,Nicholas G Brown,Anthony M Barsotti,Andrew W Stamford,Jon L Collins,Derek J Wilson,Brian Raught,Jonathan D Licht,Lindsey I James,Cheryl H Arrowsmith