日期 影响因子
日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:
–

A Novel Class of Orally Bioavailable Phenylglycine-Benzoxaborole Conjugates with Antimalarial Activity and Potentially Novel Mechanism of Action

一种新型口服生物利用度高的苯甘氨酸-苯并硼氧杂环化合物，具有抗疟活性和潜在的新型作用机制

期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.5c00549
Morake, Mokhitli; Taylor, Dale; Coertzen, Dina; Njoroge, Mathew; Krugmann, Liezl; Leshabane, Meta; da Rocha, Shanté; Qahash, Tarrick; Girling, Gareth; Coyle, Rachael; Lee, Marcus C S; Wittlin, Sergio; Llinás, Manuel; Birkholtz, Lyn-Marie; Basarab, Gregory S; Chibale, Kelly
发表日期：2026
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Negamycin: Nature's Forgotten Antibiotic

奈加霉素：被大自然遗忘的抗生素

期刊:ACS Infectious Diseases
影响因子:3.8
doi:10.1021/acsinfecdis.5c00843
Boyle, Grant A; Basarab, Gregory S
发表日期：2026
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Torque-generating units of the bacterial flagellar motor are rotary motors

细菌鞭毛马达的扭矩发生单元是旋转马达。

期刊:Proceedings of the National Academy of Sciences of the United States of America
影响因子:9.1
doi:10.1073/pnas.2515291122
Hosu, Basarab G; Vrabioiu, Alina M; Samuel, Aravinthan D T
微生物学
发表日期：2025
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Cell-Based Progression of Spiroindoline Phenotypic Hits Leads to the Identification of Compounds with Diverging Parasitological Profiles against the Human Malaria Parasite Plasmodium falciparum

基于细胞的螺吲哚啉表型先导化合物筛选，最终鉴定出针对人类疟原虫恶性疟原虫具有不同寄生虫学特征的化合物。

期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c00302
Dam, Jean; Boyle, Grant A; Horatscheck, André; Woodland, John G; Le Manach, Claire; Kaur, Gurminder; Taylor, Dale; Krugmann, Liezl; Njoroge, Mathew; Lawrence, Nina; Brunschwig, Christel; Zdorichenko, Victor; Cox, Brian; Wittlin, Sergio; von Geldern, Thomas W; Smith, Dennis; Duffy, James; Basarab, Gregory S; Chibale, Kelly
微生物学
细胞生物学
Human
发表日期：2025
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Optimization of 2,8-Diaryl-1,5-naphthyridines as Plasmodium falciparum Phosphatidylinositol 4-Kinase Inhibitors with Improved ADME Profiles and In Vivo Efficacy

优化 2,8-二芳基-1,5-萘啶类化合物作为恶性疟原虫磷脂酰肌醇 4-激酶抑制剂，以改善其 ADME 特性和体内疗效

期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c02248
Dziwornu, Godwin A; Seanego, Donald; Fienberg, Stephen; Sypu, Venkata S; Salomane, Nicolaas; Krugmann, Liezl; Taylor, Dale; Masike, Keabetswe; Njoroge, Mathew; Boonyalai, Nonlawat; Lee, Marcus C S; Godoy, Luiz C; Pasaje, Charisse Flerida; Niles, Jacquin C; Basarab, Gregory S; Coulson, Lauren B; Ghorpade, Sandeep R; Chibale, Kelly
信号转导
发表日期：2025
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Design of Novel Mercapto-3-phenylpropanoyl Dipeptides as Dual Angiotensin-Converting Enzyme C-Domain-Selective/Neprilysin Inhibitors.

设计新型巯基-3-苯基丙酰二肽作为双重血管紧张素转换酶C结构域选择性/脑啡肽酶抑制剂

期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c00329
Cozier Gyles E, Coulson Lauren B, Eyermann Charles J, Basarab Gregory S, Schwager Sylva L, Chibale Kelly, Sturrock Edward D, Acharya K Ravi
其它
血管生成
发表日期：2025
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Dose-fractionation studies of a Plasmodium phosphatidylinositol 4-kinase inhibitor in a humanized mouse model of malaria

在人源化小鼠疟疾模型中对疟原虫磷脂酰肌醇 4-激酶抑制剂进行剂量分割研究

期刊:Antimicrobial Agents and Chemotherapy
影响因子:4.5
doi:10.1128/aac.00842-24
Gibhard, Liezl; Njoroge, Mathew; Mulubwa, Mwila; Lawrence, Nina; Smith, Dennis; Duffy, James; Le Manach, Claire; Brunschwig, Christel; Taylor, Dale; van der Westhuyzen, Renier; Street, Leslie J; Basarab, Gregory S; Chibale, Kelly
微生物学
信号转导
疟疾
发表日期：2024
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Interactions between Zoliflodacin and Neisseria gonorrhoeae Gyrase and Topoisomerase IV: Enzymological Basis for Cellular Targeting

佐利氟达辛与淋病奈瑟菌DNA促旋酶和拓扑异构酶IV的相互作用：细胞靶向的酶学基础

期刊:ACS Infectious Diseases
影响因子:3.8
doi:10.1021/acsinfecdis.4c00438
Collins, Jessica A; Basarab, Gregory S; Chibale, Kelly; Osheroff, Neil
微生物学
淋病
细胞生物学
发表日期：2024
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Impact of war-associated factors on spread of sexually transmitted infections: a systemic review

战争相关因素对性传播感染扩散的影响：系统性综述

期刊:Frontiers in Public Health
影响因子:3.4
doi:10.3389/fpubh.2024.1366600
Kvasnevska, Yulia; Faustova, Mariia; Voronova, Kseniia; Basarab, Yaroslav; Lopatina, Yaroslava
炎症/感染
发表日期：2024
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"We need to talk about it, test it, prevent it, and that is our job": qualitative report on the awareness of primary care physicians regarding HIV in Ukraine

“我们需要谈论它、检测它、预防它，这是我们的职责”：乌克兰基层医生对艾滋病毒认知情况的定性报告

期刊:
影响因子:
doi:10.3389/frhs.2024.1444575
Kvasnevska, Yulia; Faustova, Mariia; Voronova, Kseniia; Basarab, Yaroslav; Lopatina, Yaroslava
HIV
神经科学
微生物学
发表日期：2024
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