日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Large Library Docking for Polypharmacology

用于多药理学的大型库对接

Wu, Yujin; Vigneron, Seth; Braz, Joao; Srinivasan, Karthik; Fink, Elissa A; Huang, Xi-Ping; Xu, Xinyu; Huebner, Harald; Kim, Joseph Y; Wang, Jing; Pfeiffer, Tara; Sakamoto, Kensuke; Radchenko, Dmytro S; Rodriguiz, Ramona M; Moroz, Yurii S; Irwin, John J; Gmeiner, Peter; Billesboelle, Christian; Roth, Bryan L; Basbaum, Allan I; Manglik, Aashish; Wetsel, William C; Shoichet, Brian K

Blood Flow Restriction Therapy Stimulates Intercellular Mitochondria Transfer and Improves Muscle Regeneration and Shoulder Function in a Murine Rotator Cuff Injury Model.

血流限制疗法可刺激细胞间线粒体转移,改善小鼠肩袖损伤模型中的肌肉再生和肩关节功能。

Milan Nesa, Wague Aboubacar, Sang Luke, Youn Alex, Sadjadi Ryan, Samimi Yusef, Montenegro Cristhian, Lizarraga Miguel, Lau Justin, Basbaum Allan I, Davies Michael R, Kim Hubert T, Feeley Brian T, Weinrich Jarret A P, Liu Xuhui

Virtual library docking for cannabinoid-1 receptor agonists with reduced side effects.

针对副作用较小的 1 型大麻素受体激动剂的虚拟库对接

Tummino Tia A, Iliopoulos-Tsoutsouvas Christos, Braz Joao M, O'Brien Evan S, Stein Reed M, Craik Veronica, Tran Ngan K, Ganapathy Suthakar, Liu Fangyu, Shiimura Yuki, Tong Fei, Ho Thanh C, Radchenko Dmytro S, Moroz Yurii S, Rosado Sian Rodriguez, Bhardwaj Karnika, Benitez Jorge, Liu Yongfeng, Kandasamy Herthana, Normand Claire, Semache Meriem, Sabbagh Laurent, Glenn Isabella, Irwin John J, Kumar Kaavya Krishna, Makriyannis Alexandros, Basbaum Allan I, Shoichet Brian K

Discovery of a functionally selective serotonin receptor (5-HT(1A)R) agonist for the treatment of pain.

发现一种功能选择性血清素受体(5-HT(1A)R)激动剂用于治疗疼痛

Ullrich Annika, Schneider Johannes, Braz João M, Neu Eduard, Staffen Nico, Stanek Markus, Bláhová Jana, Hove Tamsanqa, Albert Tamara, Allikalt Anni, Löber Stefan, Bhardwaj Karnika, Rodriguez-Rosado Sian, Fink Elissa, Rasmussen Tim, Hübner Harald, Inoue Asuka, Shoichet Brian K, Basbaum Allan I, Böttcher Bettina, Weikert Dorothee, Gmeiner Peter

Docking 14 Million Virtual Isoquinuclidines against the μ and κ Opioid Receptors Reveals Dual Antagonists-Inverse Agonists with Reduced Withdrawal Effects

将 1400 万个虚拟异喹啉类化合物与 μ 和 κ 阿片受体对接,揭示了具有降低戒断反应的双重拮抗剂-反向激动剂。

Vigneron, Seth F; Ohno, Shohei; Braz, Joao; Kim, Joseph Y; Kweon, Oh Sang; Webb, Chase; Billesbølle, Christian B; Srinivasan, Karthik; Bhardwaj, Karnika; Irwin, John J; Manglik, Aashish; Basbaum, Allan I; Ellman, Jonathan A; Shoichet, Brian K

Keratinocyte-TRPV1 sensory neuron interactions in a genetically controllable mouse model of chronic neuropathic itch.

在基因可控的慢性神经性瘙痒小鼠模型中,角质形成细胞-TRPV1感觉神经元相互作用

Crowther Andrew J, Kashem Sakeen W, Jewell Madison E, Le Chang Henry, Midavaine Élora, Rosa Casillas Mariela, Danchine Veronika, Rodriguez Sian, Kania Artur, Chen Ritchie, Braz Joao M, Basbaum Allan I

A bad break: mechanisms and assessment of acute and chronic pain after bone fracture

糟糕的骨折:骨折后急性和慢性疼痛的机制和评估

Nishimura, Haruki; Layne, Jonathan; Yamaura, Kohei; Marcucio, Ralph; Morioka, Kazuhito; Basbaum, Allan I; Weinrich, Jarret A P; Bahney, Chelsea S

Rostral ventral medulla circuits regulate both the sensory and affective dimensions of neuropathic pain: a commentary on Dogrul et al

延髓腹侧前部回路调节神经性疼痛的感觉和情感维度:对 Dogrul 等人的研究的评论

Rosa-Casillas, Mariela; Basbaum, Allan I

Deep behavioral phenotyping tracks functional recovery following tibia fracture in mice

深度行为表型分析追踪小鼠胫骨骨折后的功能恢复情况

Layne, Jonathan E; Snapper, Dustin M; Czachor, Molly E; Lam, Charles; Matityahu, Jacob D; Lind, Dane R G; Huard, Matthieu; Huard, Johnny; Morioka, Kazuhito; Motzkin, Julian C; Basbaum, Allan I; Weinrich, Jarret A P; Bahney, Chelsea S

Differential contribution of α2δ auxiliary subunits of voltage-gated calcium channels in mouse models of pain and itch

电压门控钙通道α2δ辅助亚基在小鼠疼痛和瘙痒模型中的差异性作用

Braz, Joao M; Jewell, Madison; Bhardwaj, Karnika; Rodriguez-Rosado, Sian; Craik, Veronica; Basbaum, Allan I