日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Substrate-Guided Development of HDAC11-Selective Inhibitors Featuring α‑Amino Amide Zinc-Binding Groups

基于底物导向的HDAC11选择性抑制剂的开发,该抑制剂具有α-氨基酰胺锌结合基团

Hilscher, Sebastian; Meleshin, Marat; Baselious, Fady; Barinka, Cyril; Sippl, Wolfgang; Schutkowski, Mike; Schiene-Fischer, Cordelia

Development of Fragment-Based Inhibitors of the Bacterial Deacetylase LpxC with Low Nanomolar Activity

开发低纳摩尔活性的细菌脱乙酰酶 LpxC 的片段型抑制剂

Sebastian Mielniczuk, Katharina Hoff, Fady Baselious, Yunqi Li, Jörg Haupenthal, Andreas M Kany, Maria Riedner, Holger Rohde, Katharina Rox, Anna K H Hirsch, Isabelle Krimm, Wolfgang Sippl, Ralph Holl

Comparative Structure-Based Virtual Screening Utilizing Optimized AlphaFold Model Identifies Selective HDAC11 Inhibitor

利用优化的AlphaFold模型进行基于结构的比较虚拟筛选,鉴定出选择性HDAC11抑制剂

Baselious, Fady; Hilscher, Sebastian; Robaa, Dina; Barinka, Cyril; Schutkowski, Mike; Sippl, Wolfgang