日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of [1,2,4]triazolo[1,5-a]pyrimidine-Imatinib Hybrids With Selective Cytotoxic Activity: A Mechanistically Divergent Series From Direct BCR-ABL1 Inhibition

发现具有选择性细胞毒活性的[1,2,4]三唑并[1,5-a]嘧啶-伊马替尼杂合物:与直接抑制BCR-ABL1机制不同的系列

Moura, Stefany Castro Bazan; de Oliveira, Andressa Paula; Neto, Joao de Mello Rezende; Dantas, Rafael Ferreira; Silva-Jr, Floriano Paes; Pimentel, Luiz Claudio; Carvalho, Mayara Salles do Nascimento; Leite, Debora Inacio; da Silva, Daiane Vitoria; Bastos, Monica Macedo; Boechat, Nubia

A Review on Medicinal Chemistry and Biological Activity of Dihydropyrimidinones Against HIV

二氢嘧啶酮类药物的药物化学及抗HIV生物活性研究综述

Leite, Debora I; Macedo, Fernando B; Lima, Murilo Marinho de C; Brum, Isabelle S; Oliveira, Jonathan Fragoso Miranda de; Costa, Ana Clara S; Duarte, Stella C; Moon, Sarah; Moura, Stefany de Castro B; Oliveira, Andressa P de; Boechat, Nubia; Bastos, Monica M

Ponatinib: A Review of the History of Medicinal Chemistry behind Its Development

帕纳替尼:其研发背后的药物化学史回顾

Nascimento, Mayara; Moura, Stefany; Parra, Lidia; Vasconcellos, Valeska; Costa, Gabriela; Leite, Debora; Dias, Maria; Fernandes, Tácio Vinício Amorim; Hoelz, Lucas; Pimentel, Luiz; Bastos, Monica; Boechat, Nubia

A Review of the Development of Multitarget Molecules against HIV-TB Coinfection Pathogens

针对HIV-TB合并感染病原体的多靶点分子研发进展综述

Leite, Debora Inacio; de Castro Bazan Moura, Stefany; da Conceição Avelino Dias, Maria; Costa, Carolina Catta Preta; Machado, Gustavo Peixoto; Pimentel, Luiz Claudio Ferreira; Branco, Frederico Silva Castelo; Moreira, Rui; Bastos, Monica Macedo; Boechat, Nubia

Differential plasticity and fate of brain-resident and recruited macrophages during the onset and resolution of neuroinflammation

神经炎症发生和消退过程中脑内驻留和募集巨噬细胞的差异可塑性和命运

Karen De Vlaminck, Hannah Van Hove, Daliya Kancheva, Isabelle Scheyltjens, Ana Rita Pombo Antunes, Jonathan Bastos, Monica Vara-Perez, Leen Ali, Myrthe Mampay, Lauren Deneyer, Juliana Fabiani Miranda, Ruiyao Cai, Luc Bouwens, Dimitri De Bundel, Guy Caljon, Benoît Stijlemans, Ann Massie, Jo A Van Gin

The Use of Zidovudine Pharmacophore in Multi-Target-Directed Ligands for AIDS Therapy

齐多夫定药效团在多靶点导向配体治疗艾滋病中的应用

Bianco, Maria da Conceição Avelino Dias; Inacio Leite, Debora; Silva Castelo Branco, Frederico; Boechat, Nubia; Uliassi, Elisa; Bolognesi, Maria Laura; Bastos, Monica Macedo

New Imatinib Derivatives with Antiproliferative Activity against A549 and K562 Cancer Cells.

具有抗A549和K562癌细胞增殖活性的新型伊马替尼衍生物

Oliveira Andressa, Moura Stefany, Pimentel Luiz, Neto João, Dantas Rafael, Silva-Jr Floriano, Bastos Monica, Boechat Nubia

Pyrroles as Privileged Scaffolds in the Search for New Potential HIV Inhibitors

吡咯作为寻找新型潜在HIV抑制剂的优势骨架

Bianco, Maria da Conceição Avelino Dias; Marinho, Debora Inacio Leite Firmino; Hoelz, Lucas Villas Boas; Bastos, Monica Macedo; Boechat, Nubia