日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Tumour specific HORMAD1 expression perturbs mitotic arrest and drives sensitivity to mitotic kinase inhibitors.

肿瘤特异性 HORMAD1 表达扰乱有丝分裂停滞,并导致对有丝分裂激酶抑制剂的敏感性。

Walker Callum, Kollarovic Gabriel, Weekes Daniel, Trendell Jennifer, Hoffmann Ricarda M, Martin Alexia, Ferro Riccardo, Navarro-Llinas Blanca, Hitchen Luke, Pardo Calvo Mercedes, Balan Nicolae, Kemp Harriet, Carroll Alexandra, Davidson Kathryn, Nath Sarmi, D'Uonno Nadja, Lu Ruifang, Starling Chris, Otten Marieke, Iakobachvili Nino, Marcozzi Chiara, Rahman Ilhan, Quist Jelmar, Yu Lu, Krastev Dragomir B, Amodeo Valeria, Roxanis Ioannis, Grigoriadis Anita, Bayliss Richard, Choudhary Jyoti, Haider Syed, Pines Jonathon, Pettitt Stephen J, Lord Christopher J, Tutt Andrew N J

Mechanism of interaction between the transactivation domain of N-myc and the DNA-binding surface of TFIIIC5

N-myc 转录激活结构域与 TFIIIC5 DNA 结合表面相互作用的机制

Leen, Eoin; Yeoh, Sharon; Sahak, Eka; Mitchell, Ellie; Wildsmith, Gemma; Batchelor, Matthew; Calabrese, Antonio N; Büchel, Gabriele; Bayliss, Richard

Bora bridges Aurora-A activation and substrate recognition of PLK1.

Bora 连接 Aurora-A 激活和 PLK1 的底物识别。

Miles Jennifer A, Batchelor Matthew, Walko Martin, Gunning Vanda, Wilson Andrew J, Wright Megan H, Bayliss Richard

NEK7 phosphorylation of cortactin modulates the migratory capacity of cells expressing EML4-ALK V3.

NEK7 对 cortactin 的磷酸化调节表达 EML4-ALK V3 的细胞的迁移能力。

Richardson Emily L, Knebel Axel, Straatman Kees R, Gourlay Robert, Lamont Douglas, Hardy Tara, Turnbull Robert E, Robinson Susan W, O'Regan Laura, Bayliss Richard, Fry Andrew M

High-throughput discovery and characterisation of pentafluorobenzene sulfonamide modifiers of Aurora A kinase

利用高通量方法发现和表征Aurora A激酶的五氟苯磺酰胺修饰剂

Chesti, Julian; Miles, Jennifer A; Collins, Lawrence J; McCallum, Hamish A; Foglizzo, Martina; Ahangar, Mohd Syed; Zeqiraj, Elton; Bayliss, Richard; Warriner, Stuart L; Wright, Megan H; Nelson, Adam

Covalent Peptide-Based N-Myc/Aurora-A Inhibitors Bearing Sulfonyl Fluoride Warheads

带有磺酰氟反应基团的共价肽基N-Myc/Aurora-A抑制剂

Dawber, Robert S; Gimenez, Diana; Preston, George W; Wright, Megan H; Bayliss, Richard; Warriner, Stuart L; Wilson, Andrew J

RAF inhibitors activate the integrated stress response by direct activation of GCN2

RAF抑制剂通过直接激活GCN2来激活整合应激反应。

Gilley, Rebecca; Kidger, Andrew M; Neill, Graham; Morrison, Eve; Severson, Paul; Byrne, Dominic P; Kenneth, Niall S; Bollag, Gideon; Zhang, Chao; Maia de Oliveira, Taiana; Eyers, Patrick A; Bayliss, Richard; Masson, Glenn R; Cook, Simon J

Gluebodies Offer a Route To Improve Crystal Reliability and Diversity through Transferable Nanobody Mutations That Introduce Constitutive Close Contacts

胶体提供了一种通过可转移的纳米抗体突变来提高晶体可靠性和多样性的途径,这些突变引入了组成性的紧密接触。

Ye, Mingda; Makola, Mpho; Richards, Mark W; Newman, Joseph A; Fairhead, Michael; Burgess, Selena G; Wu, Zhihuang; Maclean, Elizabeth; Wright, Nathan D; Koekemoer, Lizbé; Thompson, Andrew; Bezerra, Gustavo Arruda; Yi, Gangshun; Li, Huanyu; Rangel, Victor L; Mamalis, Dimitrios; Aitkenhead, Hazel; Davis, Benjamin G; Gilbert, Robert J C; Duerr, Katharina L; Bayliss, Richard; Gileadi, Opher; von Delft, Frank

Structural characterization and inhibition of the interaction between ch-TOG and TACC3.

ch-TOG 与 TACC3 相互作用的结构表征和抑制

Shelford James, Burgess Selena G, Rostkova Elena, Richards Mark W, Larocque Gabrielle, Sampson Josephina, Tiede Christian, Fielding Alistair J, Daviter Tina, Tomlinson Darren C, Calabrese Antonio N, Pfuhl Mark, Bayliss Richard, Royle Stephen J

FPHC Wellbeing Charter: The 'Whys' and 'Hows' of the Charter

FPHC福祉宪章:宪章的“缘由”和“方法”。

Morton, Sarah; Surman, Katy; Bayliss, Richard; Storey, Heather; Gray, Emma; Gant, Andrew; Morris, Alistair; Forbes, Anna; Cowan, Stephanie; Stevenson, Elizabeth; Hardy, Pamela; Williams, Richard