日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

New Multiparameter Index Is a Strong Predictor of Oral Bioavailability for Heterobifunctional Degraders

新型多参数指数是异双功能降解剂口服生物利用度的强预测因子

Baylon, Javier L; Chalkley, Matthew J; Siu, Tony; Shou, Wilson; Sun, Yongnian; Cai, Xianmei; Paiva, Anthony; Patel, Shivani; Zvyaga, Tatyana; Weiss, Dahlia R

Balanced Permeability Index: A Multiparameter Index for Improved In Vitro Permeability

平衡渗透指数:一种用于改善体外渗透性的多参数指数

Weiss, Dahlia R; Baylon, Javier L; Evans, Ethan D; Paiva, Anthony; Everlof, Gerry; Cutrone, Jingfang; Broccatelli, Fabio

Anti-inflammatory dopamine- and serotonin-based endocannabinoid epoxides reciprocally regulate cannabinoid receptors and the TRPV1 channel

具有抗炎作用的多巴胺和血清素类内源性大麻素环氧化物相互调节大麻素受体和TRPV1通道。

Arnold, William R; Carnevale, Lauren N; Xie, Zili; Baylon, Javier L; Tajkhorshid, Emad; Hu, Hongzhen; Das, Aditi

Endothelial ERK1/2 signaling maintains integrity of the quiescent endothelium

内皮细胞ERK1/2信号通路维持静息内皮的完整性。

Ricard, Nicolas; Scott, Rizaldy P; Booth, Carmen J; Velazquez, Heino; Cilfone, Nicholas A; Baylon, Javier L; Gulcher, Jeffrey R; Quaggin, Susan E; Chittenden, Thomas W; Simons, Michael

Drug-Drug Interactions between Atorvastatin and Dronedarone Mediated by Monomeric CYP3A4

阿托伐他汀和决奈达隆之间通过单体CYP3A4介导的药物相互作用

Denisov, Ilia G; Baylon, Javier L; Grinkova, Yelena V; Tajkhorshid, Emad; Sligar, Stephen G

Dimeric structure of the uracil:proton symporter UraA provides mechanistic insights into the SLC4/23/26 transporters

尿嘧啶:质子同向转运蛋白 UraA 的二聚体结构为 SLC4/23/26 转运蛋白提供了机制方面的见解

Yu, Xinzhe; Yang, Guanghui; Yan, Chuangye; Baylon, Javier L; Jiang, Jing; Fan, He; Lu, Guifeng; Hasegawa, Kazuya; Okumura, Hideo; Wang, Tingliang; Tajkhorshid, Emad; Li, Shuo; Yan, Nieng

Asymmetric Binding and Metabolism of Polyunsaturated Fatty Acids (PUFAs) by CYP2J2 Epoxygenase.

CYP2J2环氧酶对多不饱和脂肪酸(PUFA)的不对称结合和代谢

Arnold William R, Baylon Javier L, Tajkhorshid Emad, Das Aditi

The cellular membrane as a mediator for small molecule interaction with membrane proteins

细胞膜作为小分子与膜蛋白相互作用的介质

Mayne, Christopher G; Arcario, Mark J; Mahinthichaichan, Paween; Baylon, Javier L; Vermaas, Josh V; Navidpour, Latifeh; Wen, Po-Chao; Thangapandian, Sundarapandian; Tajkhorshid, Emad

Atomic-level description of protein-lipid interactions using an accelerated membrane model

利用加速膜模型对蛋白质-脂质相互作用进行原子级描述

Baylon, Javier L; Vermaas, Josh V; Muller, Melanie P; Arcario, Mark J; Pogorelov, Taras V; Tajkhorshid, Emad

Efficient Exploration of Membrane-Associated Phenomena at Atomic Resolution

高效探索膜相关现象的原子分辨率

Vermaas, Josh V; Baylon, Javier L; Arcario, Mark J; Muller, Melanie P; Wu, Zhe; Pogorelov, Taras V; Tajkhorshid, Emad