日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of new aurone derivatives as submicromolar CK2 inhibitors

发现新型奥酮衍生物作为亚微摩尔级CK2抑制剂

Mahdysiuk, Mykhailo V; Volynets, Galyna P; Bdzhola, Volodymyr G; Bieda, Oleksandr A; Lukashov, Sergiy S; Sapelkin, Vladislav M; Karbovskyi, Leonid L; Yarmoluk, Sergiy M

Co-expression of the RPS6KB1 and PDPK1 genes for production of activated p70S6K1 using bac-to-bac baculovirus expression system

使用 bac-to-bac 杆状病毒表达系统共表达 RPS6KB1 和 PDPK1 基因以产生活性 p70S6K1

Anna Bdzhola #, Oksana Malanchuk #, Sergii Palchevskyi, Ivan Gout, Valeriy Filonenko, Alexander Zhyvoloup

Leveraging large language models for literature-driven prioritization of protein binding pockets

利用大型语言模型进行基于文献的蛋白质结合口袋优先级排序

Stratiichuk, Roman; Melnychenko, Mykola; Koleiev, Ihor; Voitsitskyi, Taras; Husak, Vladyslav; Shevchuk, Nazar; Ostrovsky, Zakhar; Bdzhola, Volodymyr; Yesylevskyy, Semen; Starosyla, Serhii; Nafiiev, Alan

Augmenting a training dataset of the generative diffusion model for molecular docking with artificial binding pockets

利用人工结合口袋扩充分子对接生成扩散模型的训练数据集

Voitsitskyi, Taras; Bdzhola, Volodymyr; Stratiichuk, Roman; Koleiev, Ihor; Ostrovsky, Zakhar; Vozniak, Volodymyr; Khropachov, Ivan; Henitsoi, Pavlo; Popryho, Leonid; Zhytar, Roman; Yesylevskyy, Semen; Nafiiev, Alan; Starosyla, Serhii

Immunofluorescent detection of protein CoAlation in mammalian cells under oxidative stress

氧化应激下哺乳动物细胞中蛋白质CoAlation的免疫荧光检测

Oksana Malanchuk, Antonina Khoruzhenko, Viktoriia Kosach, Anna Bdzhola, Dariy Bidiuk, Charlie Brett, Ivan Gout, Valeriy Filonenko

Investigating the Regulation of Ribosomal Protein S6 Kinase 1 by CoAlation

研究 CoAlation 对核糖体蛋白 S6 激酶 1 的调节

Oksana Malanchuk, Anna Bdzhola, Sergii Palchevskyi, Volodymyr Bdzhola, Peng Chai, Olivier E Pardo, Michael J Seckl, Adrija Banerjee, Sew Yeu Peak-Chew, Mark Skehel, Lalitha Guruprasad, Alexander Zhyvoloup, Ivan Gout, Valeriy Filonenko

Pharmacophore modeling, docking and molecular dynamics simulation for identification of novel human protein kinase C beta (PKCβ) inhibitors

利用药效团建模、分子对接和分子动力学模拟鉴定新型人蛋白激酶Cβ(PKCβ)抑制剂

Starosyla, Sergiy A; Volynets, Galyna P; Protopopov, Mykola V; Bdzhola, Volodymyr G; Pashevin, Denis O; Polishchuk, Valentyna O; Kozak, Taisiia O; Stroi, Dmytro O; Dosenko, Victor E; Yarmoluk, Sergiy M

Asymmetric Dimethylation of Ribosomal S6 Kinase 2 Regulates Its Cellular Localisation and Pro-Survival Function

核糖体 S6 激酶 2 的不对称二甲基化调节其细胞定位和促生存功能

Mahmoud I Khalil, Heba M Ismail, Ganna Panasyuk, Anna Bdzhola, Valeriy Filonenko, Ivan Gout, Olivier E Pardo

Discovery of novel antituberculosis agents among 3-phenyl-5-(1-phenyl-1H-[1,2,3]triazol-4-yl)-[1,2,4]oxadiazole derivatives targeting aminoacyl-tRNA synthetases

发现针对氨酰基-tRNA合成酶的3-苯基-5-(1-苯基-1H-[1,2,3]三唑-4-基)-[1,2,4]恶二唑衍生物中的新型抗结核药物

Mariia Yu Rybak, Anatoliy O Balanda, Anna P Yatsyshyna, Igor M Kotey, Sergiy A Starosyla, Volodymyr G Bdzhola, Lubov L Lukash, Sergiy M Yarmoluk, Michael A Tukalo, Galyna P Volynets

Novel isoniazid derivative as promising antituberculosis agent

新型异烟肼衍生物作为一种有前景的抗结核药物

Volynets, Galyna P; Tukalo, Michail A; Bdzhola, Volodymyr G; Derkach, Nataliia M; Gumeniuk, Mykola I; Tarnavskiy, Sergiy S; Yarmoluk, Sergiy M