日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Potent and selective SETDB1 covalent negative allosteric modulator reduces methyltransferase activity in cells

强效且选择性的 SETDB1 共价负变构调节剂可降低细胞中的甲基转移酶活性

Mélanie Uguen, Devan J Shell, Madhushika Silva, Yu Deng, Fengling Li, Magdalena M Szewczyk, Ka Yang, Yani Zhao, Michael A Stashko, Jacqueline L Norris-Drouin, Jarod M Waybright, Serap Beldar, Justin M Rectenwald, Angie L Mordant, Thomas S Webb, Laura E Herring, Cheryl H Arrowsmith, Suzanne Ackloo, S

A Target Class Ligandability Evaluation of WD40 Repeat-Containing Proteins

WD40重复序列蛋白的靶向配体结合能力评价

Ackloo, Suzanne; Li, Fengling; Szewczyk, Magda; Seitova, Almagul; Loppnau, Peter; Zeng, Hong; Xu, Jin; Ahmad, Shabbir; Arnautova, Yelena A; Baghaie, A J; Beldar, Serap; Bolotokova, Albina; Centrella, Paolo A; Chau, Irene; Clark, Matthew A; Cuozzo, John W; Dehghani-Tafti, Saba; Disch, Jeremy S; Dong, Aiping; Dumas, Antoine; Feng, Jianwen A; Ghiabi, Pegah; Gibson, Elisa; Gilmer, Justin; Goldman, Brian; Green, Stuart R; Guié, Marie-Aude; Guilinger, John P; Harms, Nathan; Herasymenko, Oleksandra; Houliston, Scott; Hutchinson, Ashley; Kearnes, Steven; Keefe, Anthony D; Kimani, Serah W; Kramer, Trevor; Kutera, Maria; Kwak, Haejin A; Lento, Cristina; Li, Yanjun; Liu, Jenny; Loup, Joachim; Machado, Raquel A C; Mulhern, Christopher J; Perveen, Sumera; Righetto, Germanna L; Riley, Patrick; Shrestha, Suman; Sigel, Eric A; Silva, Madhushika; Sintchak, Michael D; Slakman, Belinda L; Taylor, Rhys D; Thompson, James; Torng, Wen; Underkoffler, Carl; von Rechenberg, Moritz; Walsh, Ryan T; Watson, Ian; Wilson, Derek J; Wolf, Esther; Yadav, Manisha; Yazdi, Aliakbar K; Zhang, Junyi; Zhang, Ying; Santhakumar, Vijayaratnam; Edwards, Aled M; Barsyte-Lovejoy, Dalia; Schapira, Matthieu; Brown, Peter J; Halabelian, Levon; Arrowsmith, Cheryl H

Study of caspase-6 activity in aggressive HCT116 cells using methotrexate-encapsulated lactoferrin-conjugated solid lipid nanoparticles via in silico and in vitro approaches

利用甲氨蝶呤包封的乳铁蛋白偶联固体脂质纳米颗粒,通过计算机模拟和体外方法研究侵袭性HCT116细胞中caspase-6的活性。

Bhattacharya, Sankha; Shinde, Ranajit Nivrutti; Beldar, Vishal; Khan, Rehan

Efficacy and safety of eight-week therapy with Ashwagandha root extract in improvement of sexual health in healthy men: Findings of a prospective, randomized, double-blind, placebo-controlled study

一项前瞻性、随机、双盲、安慰剂对照研究结果显示,为期八周的南非醉茄根提取物疗法能够有效且安全地改善健康男性的性健康。

Mutha, Amit Shrenikraj; Mutha, Sonali Amit; Tejuja, Anupama Hem; Beldar, Amit Shashikant; Mulay, Alok Mahendra; Langade, Deepak

Assessment of the Impact of the Novel "No Sugar Day" Initiative Based on Staff and Student Feedback: A Mixed-Methods Study

基于教职工和学生反馈对新型“无糖日”倡议影响的评估:一项混合方法研究

Jawdekar, Ashwin M; Shaikh, Anam; Basu, Anusree; Dhonde, Shivani; Neelkanthan, Shreyas; Beldar, Tejal L

Success of pulpotomy with MTA in primary teeth: A systematic review and meta-analysis

MTA在乳牙牙髓切断术中的成功率:系统评价和荟萃分析

Beldar, Tejal Laxman; Jawdekar, Ashwin Muralidhar; Mistry, Laresh Naresh

Cdyl Deficiency Brakes Neuronal Excitability and Nociception through Promoting Kcnb1 Transcription in Peripheral Sensory Neurons

Cdyl 缺乏通过促进外周感觉神经元中的 Kcnb1 转录来抑制神经元兴奋性和痛觉

Zhao-Wei Sun, Jarod M Waybright, Serap Beldar, Lu Chen, Caroline A Foley, Jacqueline L Norris-Drouin, Tian-Jie Lyu, Aiping Dong, Jinrong Min, Yu-Pu Wang, Lindsey I James, Yun Wang

Advances in polymer based Friedlander quinoline synthesis

基于聚合物的弗里德兰德喹啉合成方法的进展

Patil, Rajendra; Chavan, Jagdish; Patel, Shivnath; Beldar, Anil

PGE1 and PGA1 bind to Nurr1 and activate its transcriptional function

PGE1 和 PGA1 与 Nurr1 结合并激活其转录功能

Sreekanth Rajan #, Yongwoo Jang #, Chun-Hyung Kim #, Woori Kim #, Hui Ting Toh, Jeha Jeon, Bin Song, Aida Serra, Julien Lescar, Jun Yeob Yoo, Serap Beldar, Hong Ye, Congbao Kang, Xue-Wei Liu, Melissa Feitosa, Yeahan Kim, Dabin Hwang, Geraldine Goh, Kah-Leong Lim, Hye Min Park, Choong Hwan Lee, Sungw

Author Correction: Sequence specificity analysis of the SETD2 protein lysine methyltransferase and discovery of a SETD2 super-substrate

作者更正:SETD2蛋白赖氨酸甲基转移酶的序列特异性分析及SETD2超底物的发现

Schuhmacher, Maren Kirstin; Beldar, Serap; Khella, Mina S; Bröhm, Alexander; Ludwig, Jan; Tempel, Wolfram; Weirich, Sara; Min, Jinrong; Jeltsch, Albert