Conformation-Selective Analogues of Dasatinib Reveal Insight into Kinase Inhibitor Binding and Selectivity
达沙替尼的构象选择性类似物揭示了激酶抑制剂的结合和选择性
期刊:ACS Chemical Biology
影响因子:3.8
doi:10.1021/acschembio.5b01018
Kwarcinski, Frank E; Brandvold, Kristoffer R; Phadke, Sameer; Beleh, Omar M; Johnson, Taylor K; Meagher, Jennifer L; Seeliger, Markus A; Stuckey, Jeanne A; Soellner, Matthew B