日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Late-stage peptide modification with salicylaldehyde tag enhances affinity for nuclear factor-kappa B essential modulator

后期肽修饰用水杨醛标签增强了对核因子-κB必需调节剂的亲和力

Mason, Mattia; Peqini, Kaliroi; Uggeri, Federico; Rondelli, Diego; Sattin, Sara; Pignataro, Luca; Pellegrino, Sara; Belvisi, Laura; Scarpa, Edoardo; Bucci, Raffaella; Dal Corso, Alberto

Toward Dual-Target Glycomimetics against Two Bacterial Lectins to Fight Pseudomonas aeruginosa-Burkholderia cenocepacia Infections: A Biophysical Study

针对两种细菌凝集素的双靶点糖模拟物对抗铜绿假单胞菌-洋葱伯克霍尔德菌感染:一项生物物理学研究

Antonini, Giulia; Fares, Mario; Hauck, Dirk; Mała, Patrycja; Gillon, Emilie; Belvisi, Laura; Bernardi, Anna; Titz, Alexander; Varrot, Annabelle; Mazzotta, Sarah

Increasing the Chemical Space of L-SIGN Specific Glycomimetics

扩大L-SIGN特异性糖模拟物的化学空间

Cavazzoli, Gianluca; Delaunay, Clara; Pollastri, Sara; Panzeri, Andrea; Sattin, Sara; Thépaut, Michel; Belvisi, Laura; Fieschi, Franck; Bernardi, Anna

Antifibrotic Efficacy of a Nintedanib-Peptide Conjugate and Diagnostic Potential of a Fluorescent Companion Probe Targeting α(V)β(6) Integrin in Idiopathic Pulmonary Fibrosis

尼达尼布-肽偶联物的抗纤维化疗效及靶向α(V)β(6)整合素的荧光伴随探针在特发性肺纤维化中的诊断潜力

Bugatti, Kelly; Ferrini, Erica; Restori, Margherita; Bonfini, Costanza; Marchese, Melissa; Bianchini, Francesca; Tomassetti, Sara; Maurizio, Andrea; Baiula, Monica; Battistini, Lucia; Marcantonio, Enrico; Curti, Claudio; Civera, Monica; Belvisi, Laura; Sartori, Andrea; Stellari, Franco F; Zanardi, Franca

Unprecedented selectivity for homologous lectin targets: differential targeting of the viral receptors L-SIGN and DC-SIGN

对同源凝集素靶标前所未有的选择性:对病毒受体 L-SIGN 和 DC-SIGN 的差异性靶向

Delaunay, Clara; Pollastri, Sara; Thépaut, Michel; Cavazzoli, Gianluca; Belvisi, Laura; Bouchikri, Clémentine; Labiod, Nuria; Lasala, Fatima; Gimeno, Ana; Franconetti, Antonio; Jiménez-Barbero, Jesús; Ardá, Ana; Delgado, Rafael; Bernardi, Anna; Fieschi, Franck

A combined fragment-based virtual screening and STD-NMR approach for the identification of E-cadherin ligands

一种结合基于片段的虚拟筛选和STD-NMR的E-钙黏蛋白配体鉴定方法

Vasile, Francesca; Lavore, Francesca; Gazzola, Silvia; Vettraino, Chiara; Parisini, Emilio; Piarulli, Umberto; Belvisi, Laura; Civera, Monica

Advanced Pyrrolidine-Carbamate Self-Immolative Spacer with Tertiary Amine Handle Induces Superfast Cyclative Drug Release

具有叔胺基团的先进吡咯烷-氨基甲酸酯自毁间隔基可诱导超快速循环药物释放

Dal Corso, Alberto; Frigoli, Margaux; Prevosti, Martina; Mason, Mattia; Bucci, Raffaella; Belvisi, Laura; Pignataro, Luca; Gennari, Cesare

Rational Design of Antiangiogenic Helical Oligopeptides Targeting the Vascular Endothelial Growth Factor Receptors

靶向血管内皮生长因子受体的抗血管生成螺旋寡肽的合理设计

Zanella, Simone; Bocchinfuso, Gianfranco; De Zotti, Marta; Arosio, Daniela; Marino, Franca; Raniolo, Stefano; Pignataro, Luca; Sacco, Giovanni; Palleschi, Antonio; Siano, Alvaro S; Piarulli, Umberto; Belvisi, Laura; Formaggio, Fernando; Gennari, Cesare; Stella, Lorenzo

Neutrophil Elastase Promotes Linker Cleavage and Paclitaxel Release from an Integrin-Targeted Conjugate

中性粒细胞弹性蛋白酶促进连接子裂解和紫杉醇从整合素靶向缀合物中释放

Raposo Moreira Dias, André; Pina, Arianna; Dean, Amelia; Lerchen, Hans-Georg; Caruso, Michele; Gasparri, Fabio; Fraietta, Ivan; Troiani, Sonia; Arosio, Daniela; Belvisi, Laura; Pignataro, Luca; Dal Corso, Alberto; Gennari, Cesare

Synthesis and Biological Evaluation of RGD and isoDGR-Monomethyl Auristatin Conjugates Targeting Integrin α(V) β(3)

靶向整合素α(V)β(3)的RGD和isoDGR-单甲基奥瑞他汀缀合物的合成和生物学评价

Raposo Moreira Dias, André; Bodero, Lizeth; Martins, Ana; Arosio, Daniela; Gazzola, Silvia; Belvisi, Laura; Pignataro, Luca; Steinkühler, Christian; Dal Corso, Alberto; Gennari, Cesare; Piarulli, Umberto