Characterizing and Overriding the Structural Mechanism of the Quizartinib-Resistant FLT3 "Gatekeeper" F691L Mutation with PLX3397
使用 PLX3397 表征和克服 Quizartinib 耐药 FLT3“守门人”F691L 突变的结构机制
期刊:Cancer Discovery
影响因子:29.7
doi:10.1158/2159-8290.CD-15-0060
Catherine C Smith, Chao Zhang, Kimberly C Lin, Elisabeth A Lasater, Ying Zhang, Evan Massi, Lauren E Damon, Matthew Pendleton, Ali Bashir, Robert Sebra, Alexander Perl, Andrew Kasarskis, Rafe Shellooe, Garson Tsang, Heidi Carias, Ben Powell, Elizabeth A Burton, Bernice Matusow, Jiazhong Zhang, Wayne