Endothelial-protective effects of a G-protein-biased sphingosine-1 phosphate receptor-1 agonist, SAR247799, in type-2 diabetes rats and a randomized placebo-controlled patient trial
SAR247799 是一种 G 蛋白偏向性鞘氨醇-1-磷酸受体-1 激动剂,其在 2 型糖尿病大鼠和一项随机安慰剂对照患者试验中表现出内皮保护作用。
期刊:British Journal of Clinical Pharmacology
影响因子:3
doi:10.1111/bcp.14632
Bergougnan, Luc; Andersen, Grit; Plum-Mörschel, Leona; Evaristi, Maria Francesca; Poirier, Bruno; Tardat, Agnes; Ermer, Marcel; Herbrand, Theresa; Arrubla, Jorge; Coester, Hans Veit; Sansone, Roberto; Heiss, Christian; Vitse, Olivier; Hurbin, Fabrice; Boiron, Rania; Benain, Xavier; Radzik, David; Janiak, Philip; Muslin, Anthony J; Hovsepian, Lionel; Kirkesseli, Stephane; Deutsch, Paul; Parkar, Ashfaq A