日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A B7-H4-Targeting Antibody-Drug Conjugate Shows Antitumor Activity in PARPi and Platinum-Resistant Cancers with B7-H4 Expression

靶向 B7-H4 的抗体-药物偶联物在 PARPi 和具有 B7-H4 表达的铂耐药癌症中表现出抗肿瘤活性

Sarah B Gitto #, Margaret Whicker #, Gareth Davies #, Sushil Kumar, Krista Kinneer, Haineng Xu, Arthur Lewis, Srinivas Mamidi, Sergey Medvedev, Hyoung Kim, Judith Anderton, E Jessica Tang, Benjamin Ferman, Steven Coats, Robert W Wilkinson, Eric Brown, Daniel J Powell Jr, Fiona Simpkins

Dual blockade of BRD4 and ATR/WEE1 pathways exploits ARID1A loss in clear cell ovarian cancer

BRD4 和 ATR/WEE1 通路的双重阻断可利用透明细胞卵巢癌中的 ARID1A 缺失

Yasuto Kinose, Haineng Xu, Hyoung Kim, Sushil Kumar, Xiaoyin Shan, Erin George, Xiaolei Wang, Sergey Medvedev, Benjamin Ferman, Sarah B Gitto, Margaret Whicker, Kurt D'Andrea, Bradley Wubbenhorst, Dorothy Hallberg, Mark O'Connor, Lauren E Schwartz, Wei-Ting Hwang, Katherine L Nathanson, Gordon B Mil

CCNE1 copy number is a biomarker for response to combination WEE1-ATR inhibition in ovarian and endometrial cancer models

CCNE1 拷贝数是卵巢癌和子宫内膜癌模型中对 WEE1-ATR 联合抑制反应的生物标志物

Haineng Xu, Erin George, Yasuto Kinose, Hyoung Kim, Jennifer B Shah, Jasmine D Peake, Benjamin Ferman, Sergey Medvedev, Thomas Murtha, Carter J Barger, Kyle M Devins, Kurt D'Andrea, Bradley Wubbenhorst, Lauren E Schwartz, Wei-Ting Hwang, Gordon B Mills, Katherine L Nathanson, Adam R Karpf, Ronny Dra