First Synthesis of Racemic Trans Propargylamino-Donepezil, a Pleiotrope Agent Able to Both Inhibit AChE and MAO-B, with Potential Interest against Alzheimer's Disease
首次合成外消旋反式炔丙基氨基多奈哌齐,这是一种能够同时抑制 AChE 和 MAO-B 的多效药物,具有治疗阿尔茨海默病的潜在潜力
期刊:Molecules
影响因子:4.2
doi:10.3390/molecules26010080
Benjamin Guieu, Cedric Lecoutey, Rémi Legay, Audrey Davis, Jana Sopkova de Oliveira Santos, Cosimo Damiano Altomare, Marco Catto, Christophe Rochais, Patrick Dallemagne