日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Biophysical fragment screening of the β1-adrenergic receptor: identification of high affinity arylpiperazine leads using structure-based drug design

β1-肾上腺素受体的生物物理片段筛选:使用基于结构的药物设计鉴定高亲和力芳基哌嗪先导化合物

John A Christopher, Jason Brown, Andrew S Doré, James C Errey, Markus Koglin, Fiona H Marshall, David G Myszka, Rebecca L Rich, Christopher G Tate, Benjamin Tehan, Tony Warne, Miles Congreve

Discovery of 1,2,4-triazine derivatives as adenosine A(2A) antagonists using structure based drug design

利用基于结构的药物设计发现 1,2,4-三嗪衍生物作为腺苷 A(2A) 拮抗剂

Miles Congreve, Stephen P Andrews, Andrew S Doré, Kaspar Hollenstein, Edward Hurrell, Christopher J Langmead, Jonathan S Mason, Irene W Ng, Benjamin Tehan, Andrei Zhukov, Malcolm Weir, Fiona H Marshall

Biophysical mapping of the adenosine A2A receptor

腺苷A2A受体的生物物理映射

Andrei Zhukov, Stephen P Andrews, James C Errey, Nathan Robertson, Benjamin Tehan, Jonathan S Mason, Fiona H Marshall, Malcolm Weir, Miles Congreve