日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A self-immolative Kdn-glycoside substrate enables high-throughput screening for inhibitors of Kdnases

一种自毁型Kdn-糖苷底物可用于高通量筛选Kdn酶抑制剂。

Nejatie, Ali; Proceviat, Cameron; Gros, Christina; Steves, Elizabeth; Moore, Margo M; Vocadlo, David J; Bennet, Andrew J

An organic proton cage that is ultra-resistant to hydroxide-promoted degradation

一种对氢氧化物促进的降解具有超强抵抗力的有机质子笼

Radford, Chase L; Saatkamp, Torben; Bennet, Andrew J; Holdcroft, Steven

Development of Tunable Mechanism-Based Carbasugar Ligands that Stabilize Glycoside Hydrolases through the Formation of Transient Covalent Intermediates

开发可通过形成瞬态共价中间体稳定糖苷水解酶的可调控机制型碳糖配体

Bhosale, Sandeep; Kandalkar, Sachin; Gilormini, Pierre-André; Akintola, Oluwafemi; Rowland, Rhianna; Adabala, Pal John Pal; King, Dustin; Deen, Matthew C; Chen, Xi; Davies, Gideon J; Vocadlo, David J; Bennet, Andrew J

Mechanism-Based Allylic Carbasugar Chlorides That Form Covalent Intermediates with α- and β-Galactosidases

能与α-和β-半乳糖苷酶形成共价中间体的基于机制的烯丙基碳糖氯化物

Akintola, Oluwafemi; Bhosale, Sandeep; Bennet, Andrew J

A heme•DNAzyme activated by hydrogen peroxide catalytically oxidizes thioethers by direct oxygen atom transfer rather than by a Compound I-like intermediate

过氧化氢激活的血红素•DNA酶通过直接氧原子转移而非类似化合物I的中间体催化氧化硫醚。

Shumayrikh, Nisreen M; Warren, Jeffrey J; Bennet, Andrew J; Sen, Dipankar

An Epoxide Intermediate in Glycosidase Catalysis

糖苷酶催化中的环氧化物中间体

Sobala, Lukasz F; Speciale, Gaetano; Zhu, Sha; Raich, Lluís; Sannikova, Natalia; Thompson, Andrew J; Hakki, Zalihe; Lu, Dan; Shamsi Kazem Abadi, Saeideh; Lewis, Andrew R; Rojas-Cervellera, Víctor; Bernardo-Seisdedos, Ganeko; Zhang, Yongmin; Millet, Oscar; Jiménez-Barbero, Jesús; Bennet, Andrew J; Sollogoub, Matthieu; Rovira, Carme; Davies, Gideon J; Williams, Spencer J

Author Correction: Revealing the mechanism for covalent inhibition of glycoside hydrolases by carbasugars at an atomic level

作者更正:从原子层面揭示碳水化合物对糖苷水解酶的共价抑制机制

Ren, Weiwu; Pengelly, Robert; Farren-Dai, Marco; Abadi, Saeideh Shamsi Kazem; Oehler, Verena; Akintola, Oluwafemi; Draper, Jason; Meanwell, Michael; Chakladar, Saswati; Świderek, Katarzyna; Moliner, Vicent; Britton, Robert; Gloster, Tracey M; Bennet, Andrew J

Revealing the mechanism for covalent inhibition of glycoside hydrolases by carbasugars at an atomic level.

从原子水平揭示糖苷水解酶共价抑制的机制

Ren Weiwu, Pengelly Robert, Farren-Dai Marco, Shamsi Kazem Abadi Saeideh, Oehler Verena, Akintola Oluwafemi, Draper Jason, Meanwell Michael, Chakladar Saswati, Świderek Katarzyna, Moliner Vicent, Britton Robert, Gloster Tracey M, Bennet Andrew J

Structural Snapshots for Mechanism-Based Inactivation of a Glycoside Hydrolase by Cyclopropyl Carbasugars

环丙基碳糖对糖苷水解酶机制性失活的结构快照

Adamson, Christopher; Pengelly, Robert J; Shamsi Kazem Abadi, Saeideh; Chakladar, Saswati; Draper, Jason; Britton, Robert; Gloster, Tracey M; Bennet, Andrew J

Metabolism of vertebrate amino sugars with N-glycolyl groups: intracellular β-O-linked N-glycolylglucosamine (GlcNGc), UDP-GlcNGc, and the biochemical and structural rationale for the substrate tolerance of β-O-linked β-N-acetylglucosaminidase

脊椎动物含N-羟乙酰基氨基糖的代谢:细胞内β-O-连接的N-羟乙酰氨基葡萄糖(GlcNGc)、UDP-GlcNGc,以及β-O-连接的β-N-乙酰氨基葡萄糖苷酶底物耐受性的生化和结构基础

Macauley, Matthew S; Chan, Jefferson; Zandberg, Wesley F; He, Yuan; Whitworth, Garrett E; Stubbs, Keith A; Yuzwa, Scott A; Bennet, Andrew J; Varki, Ajit; Davies, Gideon J; Vocadlo, David J