Carboxylic acid isosteres improve the activity of ring-fused 2-pyridones that inhibit pilus biogenesis in E. coli
羧酸等排体可提高环稠合2-吡啶酮的活性,该类化合物可抑制大肠杆菌菌毛的生物合成。
期刊:Bioorganic & Medicinal Chemistry Letters
影响因子:2.2
doi:10.1016/j.bmcl.2008.05.020
Berg, Veronica; Das, Pralay; Chorell, Erik; Hedenström, Mattias; Pinkner, Jerome S; Hultgren, Scott J; Almqvist, Fredrik