日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Advancing Isotope Labeling Technologies at AstraZeneca through Academic-Industrial Collaboration

阿斯利康通过产学研合作推进同位素标记技术发展

Bragg, Ryan A; Bergare, Jonas; Artelsmair, Markus; Kerr, William J; Skrydstrup, Troels; Elmore, Charles S

Efficient palladium-catalyzed electrocarboxylation enables late-stage carbon isotope labelling

高效的钯催化电羧化反应可实现后期碳同位素标记

Batista, Gabriel M F; Ebenbauer, Ruth; Day, Craig; Bergare, Jonas; Neumann, Karoline T; Hopmann, Kathrin H; Elmore, Charles S; Rosas-Hernández, Alonso; Skrydstrup, Troels

Identification and In Vitro and In Vivo Characterization of KAC-50.1 as a Potential α-Synuclein PET Radioligand

KAC-50.1作为潜在的α-突触核蛋白PET放射性配体的鉴定、体外和体内表征

Saturnino Guarino, Dinahlee; Miranda Azpiazu, Patricia; Sunnemark, Dan; Elmore, Charles S; Bergare, Jonas; Artelsmair, Markus; Nordvall, Gunnar; Forsberg Morén, Anton; Jia, Zhisheng; Cortes-Gonzalez, Miguel; Mach, Robert H; Wilcox, Kyle C; Finnema, Sjoerd; Schou, Magnus; Varrone, Andrea

Synthesis and preclinical evaluation of [11C]EAI045 as a PET tracer for imaging tumors expressing mutated epidermal growth factor receptor

[11C]EAI045 的合成及作为 PET 示踪剂对表达突变表皮生长因子受体的肿瘤进行成像的临床前评估

Antonia A Högnäsbacka, Alex J Poot, Christophe Plisson, Jonas Bergare, David R Bonsall, Stuart P McCluskey, Lisa A Wells, Esther Kooijman, Robert C Schuit, Mariska Verlaan, Wissam Beaino, Guus A M S van Dongen, Danielle J Vugts, Charles S Elmore, Jan Passchier, Albert D Windhorst

Pharmacokinetic Evaluation of New Drugs Using a Multi-Labelling Approach and PET Imaging: Application to a Drug Candidate with Potential Application in Neuromuscular Disorders

使用多标记方法和 PET 成像对新药进行药代动力学评估:应用于可能用于治疗神经肌肉疾病的候选药物

Rossana Passannante, Vanessa Gómez-Vallejo, Maialen Sagartzazu-Aizpurua, Laura Vignau Arsuaga, Pablo Marco-Moreno, Garazi Aldanondo, Ainara Vallejo-Illarramendi, Pablo Aguiar, Unai Cossío, Abraham Martín, Jonas Bergare, Lee Kingston, Charles S Elmore, Miguel Angel Morcillo, Pablo Ferrón, Jesus M Aiz

Computationally-Guided Development of a Chelated NHC-P Iridium(I) Complex for the Directed Hydrogen Isotope Exchange of Aryl Sulfones

利用计算方法开发螯合NHC-P铱(I)配合物用于芳基砜的定向氢同位素交换

Kerr, William J; Knox, Gary J; Reid, Marc; Tuttle, Tell; Bergare, Jonas; Bragg, Ryan A

Synthesis, (3) H-labelling and in vitro evaluation of a substituted dipiperidine alcohol as a potential ligand for chemokine receptor 2

(3)合成、H标记和体外评价取代的二哌啶醇作为趋化因子受体2的潜在配体

Artelsmair, Markus; Miranda-Azpiazu, Patricia; Kingston, Lee; Bergare, Jonas; Schou, Magnus; Varrone, Andrea; Elmore, Charles S

Differential Pharmacology and Binding of mGlu(2) Receptor Allosteric Modulators

mGlu(2)受体变构调节剂的差异药理学和结合

O'Brien, Daniel E; Shaw, Douglas M; Cho, Hyekyung P; Cross, Alan J; Wesolowski, Steven S; Felts, Andrew S; Bergare, Jonas; Elmore, Charles S; Lindsley, Craig W; Niswender, Colleen M; Conn, P Jeffrey