日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Exploiting the 2-(1,3,4,9-tetrahydropyrano[3,4-b]indol-1-yl)acetic Acid Scaffold to Generate COXTRANs: A New Class of Dual Cyclooxygenase Inhibitors-Thromboxane Receptor Antagonists

利用 2-(1,3,4,9-四氢吡喃并[3,4-b]吲哚-1-基)乙酸骨架生成 COXTRANs:一类新型双重环氧合酶抑制剂-血栓素受体拮抗剂

Blua, Federica; Boccato, Francesca; Buccellati, Carola; Risè, Patrizia; Barbieri, Silvia; Castiglioni, Laura; Balzulat, Annika; Rolando, Barbara; Marini, Elisabetta; Balestra, Marta; Introvigne, Maria Luisa; Giorgis, Marta; Sironi, Luigi; Tacconelli, Stefania; Hiesinger, Kerstin; Patrignani, Paola; Schmidtko, Achim; Steinhilber, Dieter; Proschak, Ewgenij; Sala, Angelo; Rovati, G Enrico; Bertinaria, Massimo

Multitarget Antioxidant NO-Donor Organic Nitrates: A Novel Approach to Overcome Nitrates Tolerance, an Ex Vivo Study

多靶点抗氧化剂NO供体有机硝酸盐:克服硝酸盐耐受性的新方法——一项离体研究

Marini, Elisabetta; Giorgis, Marta; Leporati, Marta; Rolando, Barbara; Chegaev, Konstantin; Lazzarato, Loretta; Bertinaria, Massimo; Vincenti, Marco; Di Stilo, Antonella

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-7

药物化学的突破:新靶点和机制、新药物、新希望-7

Gütschow, Michael; Eynde, Jean Jacques Vanden; Jampilek, Josef; Kang, CongBao; Mangoni, Arduino A; Fossa, Paola; Karaman, Rafik; Trabocchi, Andrea; Scott, Peter J H; Reynisson, Jóhannes; Rapposelli, Simona; Galdiero, Stefania; Winum, Jean-Yves; Brullo, Chiara; Prokai-Tatrai, Katalin; Sharma, Arun K; Schapira, Matthieu; Azuma, Yasu-Taka; Cerchia, Laura; Spetea, Mariana; Torri, Giangiacomo; Collina, Simona; Geronikaki, Athina; García-Sosa, Alfonso T; Vasconcelos, M Helena; Sousa, Maria Emília; Kosalec, Ivan; Tuccinardi, Tiziano; Duarte, Iola F; Salvador, Jorge A R; Bertinaria, Massimo; Pellecchia, Maurizio; Amato, Jussara; Rastelli, Giulio; Gomes, Paula A C; Guedes, Rita C; Sabatier, Jean-Marc; Estévez-Braun, Ana; Pagano, Bruno; Mangani, Stefano; Ragno, Rino; Kokotos, George; Brindisi, Margherita; González, Florenci V; Borges, Fernanda; Miloso, Mariarosaria; Rautio, Jarkko; Muñoz-Torrero, Diego

Ticagrelor Conditioning Effects Are Not Additive to Cardioprotection Induced by Direct NLRP3 Inflammasome Inhibition: Role of RISK, NLRP3, and Redox Cascades.

替格瑞洛的预处理作用不能叠加于直接抑制 NLRP3 炎症小体所诱导的心脏保护作用:RISK、NLRP3 和氧化还原级联的作用

Penna Claudia, Aragno Manuela, Cento Alessia Sofia, Femminò Saveria, Russo Isabella, Bello Federica Dal, Chiazza Fausto, Collotta Debora, Alves Gustavo Ferreira, Bertinaria Massimo, Zicola Elisa, Mercurio Valentina, Medana Claudio, Collino Massimo, Pagliaro Pasquale

A Comparative Study on the Efficacy of NLRP3 Inflammasome Signaling Inhibitors in a Pre-clinical Model of Bowel Inflammation

NLRP3炎症小体信号抑制剂在肠道炎症临床前模型中的疗效比较研究

Pellegrini, Carolina; Fornai, Matteo; Colucci, Rocchina; Benvenuti, Laura; D’Antongiovanni, Vanessa; Natale, Gianfranco; Fulceri, Federica; Giorgis, Marta; Marini, Elisabetta; Gastaldi, Simone; Bertinaria, Massimo; Blandizzi, Corrado; Antonioli, Luca

Pharmacological Inhibition of NLRP3 Inflammasome Attenuates Myocardial Ischemia/Reperfusion Injury by Activation of RISK and Mitochondrial Pathways

NLRP3炎症小体的药理学抑制通过激活RISK和线粒体通路减轻心肌缺血/再灌注损伤

Mastrocola, Raffaella; Penna, Claudia; Tullio, Francesca; Femminò, Saveria; Nigro, Debora; Chiazza, Fausto; Serpe, Loredana; Collotta, Debora; Alloatti, Giuseppe; Cocco, Mattia; Bertinaria, Massimo; Pagliaro, Pasquale; Aragno, Manuela; Collino, Massimo

NO-Donor Dihydroartemisinin Derivatives as Multitarget Agents for the Treatment of Cerebral Malaria

NO供体双氢青蒿素衍生物作为治疗脑型疟疾的多靶点药物

Bertinaria, Massimo; Orjuela-Sanchez, Pamela; Marini, Elisabetta; Guglielmo, Stefano; Hofer, Anthony; Martins, Yuri C; Zanini, Graziela M; Frangos, John A; Gasco, Alberto; Fruttero, Roberta; Carvalho, Leonardo J M