日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

DYRK1A inhibition results in MYC and ERK activation rendering KMT2A-R acute lymphoblastic leukemia cells sensitive to BCL2 inhibition

DYRK1A抑制导致MYC和ERK激活,使KMT2A-R急性淋巴细胞白血病细胞对BCL2抑制敏感。

Ayyadevara, V S S Abhinav; Wertheim, Gerald; Gaur, Shikha; Chukinas, John A; Loftus, Joseph P; Lee, Sung June; Kumar, Anil; Swaminathan, Srividya; Bhansali, Rahul S; Childers, Wayne; Geng, Huimin; Milne, Thomas A; Hua, Xianxin; Bernt, Kathrin M; Besson, Thierry; Shi, Junwei; Crispino, John D; Carroll, Martin; Tasian, Sarah K; Hurtz, Christian

Quinazoline-Derivatives of Imino-1,2,3-Dithiazoles Promote Biofilm Dispersion of Pseudomonas aeruginosa

亚氨基-1,2,3-二噻唑的喹唑啉衍生物促进铜绿假单胞菌生物膜的分散

Gonzalez, Mathieu; Tareau, Anne-Sophie; de Crozals, Daphnée; Layec, Corentin; Broudic, Nathan; Barreau, Magalie; Forge, Adrien; Lesouhaitier, Olivier; Fruit, Corinne; Chevalier, Sylvie; Besson, Thierry; Tahrioui, Ali

Efficacy of DYRK1A inhibitors in novel models of Down syndrome acute lymphoblastic leukemia

DYRK1A抑制剂在唐氏综合征急性淋巴细胞白血病新型模型中的疗效

Carey-Smith, Shannon L; Simad, Maryam H; Panchal, Kunjal; Aya-Bonilla, Carlos; Smolders, Hannah; Lin, Sang; Armitage, Jesse D; Nguyen, Vivien T; Bentley, Kathryn; Ford, Jette; Singh, Sajla; Oommen, Joyce; Laurent, Anouchka P; Mercher, Thomas; Crispino, John D; Montgomery, Andrew P; Kassiou, Michael; Besson, Thierry; Deau, Emmanuel; Meijer, Laurent; Cheung, Laurence C; Kotecha, Rishi S; Malinge, Sébastien

Novel Thiazole-Fused [4,5-g] or [5,4-g]Quinazolin-8-ones and Their Quinazoline Analogues: Synthesis and Biological Evaluation.

新型噻唑稠合[4,5-g]或[5,4-g]喹唑啉-8-酮及其喹唑啉类似物:合成和生物学评价

Broudic Nathan, Pacheco-Benichou Alexandra, Corbière Cécile, Baratte Blandine, Robert Thomas, Bach Stéphane, Solhi Hélène, Le Guével Rémy, Fruit Corinne, Besson Thierry

Recent Advances in Transition-Metal-Free Late-Stage C-H and N-H Arylation of Heteroarenes Using Diaryliodonium Salts

利用二芳基碘鎓盐实现杂芳烃无过渡金属后期CH和NH芳基化反应的最新进展

Besson, Thierry; Fruit, Corinne

Demonstration of Green Solvent Performance on O,S,N-Heterocycles Synthesis: Metal-Free Click Chemistry and Buchwald-Hartwig Coupling

绿色溶剂在 O,S,N-杂环化合物合成中的性能展示:无金属点击化学和 Buchwald-Hartwig 偶联反应

Campos, Joana F; Cailler, Manon; Claudel, Remi; Prot, Benjamin; Besson, Thierry; Berteina-Raboin, Sabine