日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Crystal structure of Crocus vernus class IIIb chitinase: in silico ligand-binding studies and in vitro antifungal assay

番红花IIIb类几丁质酶的晶体结构:计算机模拟配体结合研究和体外抗真菌活性测定

Saeed, Ahsan; Khaliq, Binish; Iqbal, Sadaf; Mehmood, Sohaib; Betzel, Christian; Akrem, Ahmed

Unveiling the structure, function and dynamics of StmPr1 in Stenotrophomonas maltophilia virulence

揭示嗜麦芽窄食单胞菌毒力中 StmPr1 的结构、功能和动态

Sommer, Max; Negm, Amr; Outzen, Lasse; Windhorst, Sabine; Gabdulkhakov, Azat; Weber, Wolfgang; Betzel, Christian

SARS-CoV-2 M(pro) responds to oxidation by forming disulfide and NOS/SONOS bonds

SARS-CoV-2 M(pro) 通过形成二硫键和 NOS/SONOS 键来响应氧化反应。

Reinke, Patrick Y A; Schubert, Robin; Oberthür, Dominik; Galchenkova, Marina; Rahmani Mashhour, Aida; Günther, Sebastian; Chretien, Anaïs; Round, Adam; Seychell, Brandon Charles; Norton-Baker, Brenna; Kim, Chan; Schmidt, Christina; Koua, Faisal H M; Tolstikova, Alexandra; Ewert, Wiebke; Peña Murillo, Gisel Esperanza; Mills, Grant; Kirkwood, Henry; Brognaro, Hévila; Han, Huijong; Koliyadu, Jayanath; Schulz, Joachim; Bielecki, Johan; Lieske, Julia; Maracke, Julia; Knoska, Juraj; Lorenzen, Kristina; Brings, Lea; Sikorski, Marcin; Kloos, Marco; Vakili, Mohammad; Vagovic, Patrik; Middendorf, Philipp; de Wijn, Raphael; Bean, Richard; Letrun, Romain; Han, Seonghyun; Falke, Sven; Geng, Tian; Sato, Tokushi; Srinivasan, Vasundara; Kim, Yoonhee; Yefanov, Oleksandr M; Gelisio, Luca; Beck, Tobias; Doré, Andrew S; Mancuso, Adrian P; Betzel, Christian; Bajt, Saša; Redecke, Lars; Chapman, Henry N; Meents, Alke; Turk, Dušan; Hinrichs, Winfried; Lane, Thomas J

Time-resolved crystallography of boric acid binding to the active site serine of the β-lactamase CTX-M-14 and subsequent 1,2-diol esterification

利用时间分辨晶体学方法研究硼酸与β-内酰胺酶CTX-M-14活性位点丝氨酸结合及其后续的1,2-二醇酯化反应。

Prester, Andreas; Perbandt, Markus; Galchenkova, Marina; Oberthuer, Dominik; Werner, Nadine; Henkel, Alessandra; Maracke, Julia; Yefanov, Oleksandr; Hakanpää, Johanna; Pompidor, Guillaume; Meyer, Jan; Chapman, Henry; Aepfelbacher, Martin; Hinrichs, Winfried; Rohde, Holger; Betzel, Christian

Antiviral activity of natural phenolic compounds in complex at an allosteric site of SARS-CoV-2 papain-like protease

天然酚类化合物与SARS-CoV-2木瓜蛋白酶样蛋白酶变构位点形成复合物的抗病毒活性

Srinivasan, Vasundara; Brognaro, Hévila; Prabhu, Prince R; de Souza, Edmarcia Elisa; Günther, Sebastian; Reinke, Patrick Y A; Lane, Thomas J; Ginn, Helen; Han, Huijong; Ewert, Wiebke; Sprenger, Janina; Koua, Faisal H M; Falke, Sven; Werner, Nadine; Andaleeb, Hina; Ullah, Najeeb; Franca, Bruno Alves; Wang, Mengying; Barra, Angélica Luana C; Perbandt, Markus; Schwinzer, Martin; Schmidt, Christina; Brings, Lea; Lorenzen, Kristina; Schubert, Robin; Machado, Rafael Rahal Guaragna; Candido, Erika Donizette; Oliveira, Danielle Bruna Leal; Durigon, Edison Luiz; Niebling, Stephan; Garcia, Angelica Struve; Yefanov, Oleksandr; Lieske, Julia; Gelisio, Luca; Domaracky, Martin; Middendorf, Philipp; Groessler, Michael; Trost, Fabian; Galchenkova, Marina; Mashhour, Aida Rahmani; Saouane, Sofiane; Hakanpää, Johanna; Wolf, Markus; Alai, Maria Garcia; Turk, Dusan; Pearson, Arwen R; Chapman, Henry N; Hinrichs, Winfried; Wrenger, Carsten; Meents, Alke; Betzel, Christian

Hydrazones and Thiosemicarbazones Targeting Protein-Protein-Interactions of SARS-CoV-2 Papain-like Protease

腙类和硫代氨基脲类化合物靶向SARS-CoV-2木瓜蛋白酶样蛋白酶的蛋白质-蛋白质相互作用

Ewert, Wiebke; Günther, Sebastian; Miglioli, Francesca; Falke, Sven; Reinke, Patrick Y A; Niebling, Stephan; Günther, Christian; Han, Huijong; Srinivasan, Vasundara; Brognaro, Hévila; Lieske, Julia; Lorenzen, Kristina; Garcia-Alai, Maria M; Betzel, Christian; Carcelli, Mauro; Hinrichs, Winfried; Rogolino, Dominga; Meents, Alke

Structural characterization and antibacterial activity of silver nanoparticles synthesized using a low-molecular-weight Royal Jelly extract

利用低分子量蜂王浆提取物合成银纳米粒子的结构表征及抗菌活性研究

Gevorgyan, Susanna; Schubert, Robin; Falke, Sven; Lorenzen, Kristina; Trchounian, Karen; Betzel, Christian

Structural basis to repurpose boron-based proteasome inhibitors Bortezomib and Ixazomib as β-lactamase inhibitors

将硼基蛋白酶体抑制剂硼替佐米和伊沙佐米重新用作β-内酰胺酶抑制剂的结构基础

Perbandt, Markus; Werner, Nadine; Prester, Andreas; Rohde, Holger; Aepfelbacher, Martin; Hinrichs, Winfried; Betzel, Christian

Structure and activity of the DHNA Coenzyme-A Thioesterase from Staphylococcus aureus providing insights for innovative drug development

金黄色葡萄球菌DHNA辅酶A硫酯酶的结构和活性为创新药物研发提供了见解

Murad, Aline Melro; Brognaro, Hévila; Falke, Sven; Lindner, Jasmin; Perbandt, Markus; Mudogo, Celestin; Schubert, Robin; Wrenger, Carsten; Betzel, Christian

Intrinsically disordered plant protein PARCL colocalizes with RNA in phase-separated condensates whose formation can be regulated by mutating the PLD

固有无序植物蛋白PARCL与RNA共定位于相分离凝聚体中,而这些凝聚体的形成可通过PLD突变进行调控。

Ostendorp, Anna; Ostendorp, Steffen; Zhou, Yuan; Chaudron, Zoé; Wolffram, Lukas; Rombi, Khadija; von Pein, Linn; Falke, Sven; Jeffries, Cy M; Svergun, Dmitri I; Betzel, Christian; Morris, Richard J; Kragler, Friedrich; Kehr, Julia