Translation of HDAC6 PET Imaging Using [(18)F]EKZ-001-cGMP Production and Measurement of HDAC6 Target Occupancy in Nonhuman Primates
利用[(18)F]EKZ-001-cGMP生产进行HDAC6 PET成像,并测量非人灵长类动物中HDAC6靶点占有率
期刊:ACS Chemical Neuroscience
影响因子:3.9
doi:10.1021/acschemneuro.0c00074
Celen, Sofie; Rokka, Johanna; Gilbert, Tonya M; Koole, Michel; Vermeulen, Isabeau; Serdons, Kim; Schroeder, Frederick A; Wagner, Florence F; Bleeser, Tom; Hightower, Baileigh G; Hu, Jiyun; Rahal, Dania; Beyzavi, Hudson; Vanduffel, Wim; Van Laere, Koen; Kranz, Janice E; Hooker, Jacob M; Bormans, Guy; Cawthorne, Christopher J