日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Silicon incorporated tacrine: design, synthesis, and evaluation of biological and pharmacokinetic parameters

硅掺杂他克林:设计、合成及生物学和药代动力学参数评价

Kulkarni, Akshay S; Ramana, Sreenivasa Rao; Nuthakki, Vijay K; Bhatt, Shipra; Jamwal, Ashiya; Nandawadekar, Laxman D; Jotshi, Anshika; Kumar, Ajay; Nandi, Utpal; Bharate, Sandip B; Reddy, D Srinivasa

Strategies to target SARS-CoV-2 entry and infection using dual mechanisms of inhibition by acidification inhibitors

利用酸化抑制剂的双重抑制机制靶向SARS-CoV-2入侵和感染的策略

Prabhakara, Chaitra; Godbole, Rashmi; Sil, Parijat; Jahnavi, Sowmya; Gulzar, Shah-E-Jahan; van Zanten, Thomas S; Sheth, Dhruv; Subhash, Neeraja; Chandra, Anchal; Shivaraj, Akshatha; Panikulam, Patricia; U, Ibrahim; Nuthakki, Vijay Kumar; Puthiyapurayil, Theja Parassini; Ahmed, Riyaz; Najar, Ashaq Hussain; Lingamallu, Sai Manoz; Das, Snigdhadev; Mahajan, Bhagyashri; Vemula, Praveen; Bharate, Sandip B; Singh, Parvinder Pal; Vishwakarma, Ram; Guha, Arjun; Sundaramurthy, Varadharajan; Mayor, Satyajit

Discovery of Helminthosporin, an Anthraquinone Isolated from Rumex abyssinicus Jacq as a Dual Cholinesterase Inhibitor

从深海酸模(Rumex abyssinicus Jacq)中分离得到的蒽醌类化合物Helminthosporin,被发现具有双重胆碱酯酶抑制剂活性

Augustin, Ntemafack; Nuthakki, Vijay K; Abdullaha, Mohd; Hassan, Qazi Parvaiz; Gandhi, Sumit G; Bharate, Sandip B

Preclinical Development of Crocus sativus-Based Botanical Lead IIIM-141 for Alzheimer's Disease: Chemical Standardization, Efficacy, Formulation Development, Pharmacokinetics, and Safety Pharmacology

番红花类植物先导化合物IIIM-141治疗阿尔茨海默病的临床前开发:化学标准化、疗效、制剂开发、药代动力学和安全性药理学

Bharate, Sonali S; Kumar, Vikas; Singh, Gurdarshan; Singh, Amarinder; Gupta, Mehak; Singh, Deepika; Kumar, Ajay; Vishwakarma, Ram A; Bharate, Sandip B

Biotransformation, Using Recombinant CYP450-Expressing Baker's Yeast Cells, Identifies a Novel CYP2D6.10(A122V) Variant Which Is a Superior Metabolizer of Codeine to Morphine Than the Wild-Type Enzyme.

利用重组 CYP450 表达的面包酵母细胞进行生物转化,鉴定出一种新的 CYP2D6.10(A122V) 变体,该变体比野生型酶更能有效地将可待因代谢为吗啡

Williams Ibidapo S, Gatchie Linda, Bharate Sandip B, Chaudhuri Bhabatosh

Boeravinone B, A Novel Dual Inhibitor of NorA Bacterial Efflux Pump of Staphylococcus aureus and Human P-Glycoprotein, Reduces the Biofilm Formation and Intracellular Invasion of Bacteria

Boeravinone B 是一种新型的金黄色葡萄球菌 NorA 细菌外排泵和人 P-糖蛋白双重抑制剂,可减少细菌生物膜的形成和细胞内侵袭。

Singh, Samsher; Kalia, Nitin P; Joshi, Prashant; Kumar, Ajay; Sharma, Parduman R; Kumar, Ashok; Bharate, Sandip B; Khan, Inshad A

Non-enzymatic browning in citrus juice: chemical markers, their detection and ways to improve product quality

柑橘汁非酶褐变:化学标记物、检测方法及提高产品质量的途径

Bharate, Sonali S; Bharate, Sandip B

Thionate versus Oxon: comparison of stability, uptake, and cell toxicity of ((14)CH(3)O)(2)-labeled methyl parathion and methyl paraoxon with SH-SY5Y cells

硫代磷酸酯与氧磷:(14)CH(3)O)2-标记的甲基对硫磷和甲基对氧磷对SH-SY5Y细胞的稳定性、摄取和细胞毒性比较

Bharate, Sandip B; Prins, John M; George, Kathleen M; Thompson, Charles M

Antimicrobial, antimalarial, and antileishmanial activities of mono- and bis-quaternary pyridinium compounds

单季铵和双季铵吡啶化合物的抗菌、抗疟疾和抗利什曼原虫活性

Bharate, Sandip B; Thompson, Charles M

New series of monoquaternary pyridinium oximes: Synthesis and reactivation potency for paraoxon-inhibited electric eel and recombinant human acetylcholinesterase

新型单季铵吡啶肟系列化合物:合成及其对对氧磷抑制的电鳗和重组人乙酰胆碱酯酶的再活化效力

Bharate, Sandip B; Guo, Lilu; Reeves, Tony E; Cerasoli, Douglas M; Thompson, Charles M