日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Deoxyguanosine-Linked Bifunctional Inhibitor of SAMHD1 dNTPase Activity and Nucleic Acid Binding

脱氧鸟苷连接的SAMHD1 dNTPase活性和核酸结合双功能抑制剂

Egleston, Matthew; Dong, Linghao; Howlader, A Hasan; Bhat, Shridhar; Orris, Benjamin; Bianchet, Mario A; Greenberg, Marc M; Stivers, James T

Rapamycin-inspired macrocycles with new target specificity

雷帕霉素启发的具有新型靶向特异性的大环化合物

Guo, Zufeng; Hong, Sam Y; Wang, Jingxin; Rehan, Shahid; Liu, Wukun; Peng, Hanjing; Das, Manisha; Li, Wei; Bhat, Shridhar; Peiffer, Brandon; Ullman, Brett R; Tse, Chung-Ming; Tarmakova, Zlatina; Schiene-Fischer, Cordelia; Fischer, Gunter; Coe, Imogen; Paavilainen, Ville O; Sun, Zhaoli; Liu, Jun O

Hydrazide Mimics for Protein Lysine Acylation To Assess Nucleosome Dynamics and Deubiquitinase Action

利用酰肼类似物模拟蛋白质赖氨酸酰化,以评估核小体动力学和去泛素化酶活性

Bhat, Shridhar; Hwang, Yousang; Gibson, Matthew D; Morgan, Michael T; Taverna, Sean D; Zhao, Yingming; Wolberger, Cynthia; Poirier, Michael G; Cole, Philip A

Tricyclic thiazoles are a new class of angiogenesis inhibitors

三环噻唑类化合物是一类新型血管生成抑制剂。

Bhat, Shridhar; Shim, Joong Sup; Liu, Jun O

Inhibition of eukaryotic translation elongation by the antitumor natural product Mycalamide B.

抗肿瘤天然产物Mycalamide B抑制真核翻译延伸

Dang Yongjun, Schneider-Poetsch Tilman, Eyler Daniel E, Jewett John C, Bhat Shridhar, Rawal Viresh H, Green Rachel, Liu Jun O

Diazo reagents with small steric footprints for simultaneous arming/SAR studies of alcohol-containing natural products via O-H insertion

具有小空间位阻的重氮试剂可用于通过OH插入同时对含醇天然产物进行配体修饰/构效关系研究。

Chamni, Supakarn; He, Qing-Li; Dang, Yongjun; Bhat, Shridhar; Liu, Jun O; Romo, Daniel

A simple and efficient route to the FKBP-binding domain from rapamycin

从雷帕霉素合成FKBP结合域的一种简便高效的方法

Li, Wei; Bhat, Shridhar; Liu, Jun O

Inhibition of amyloid A amyloidogenesis in vivo and in tissue culture by 4-deoxy analogues of peracetylated 2-acetamido-2-deoxy-alpha- and beta-d-glucose: implications for the treatment of various amyloidoses

4-脱氧类似物对体内和组织培养中全乙酰化2-乙酰氨基-2-脱氧-α-和β-D-葡萄糖抑制淀粉样蛋白A淀粉样变性的作用:对各种淀粉样变性治疗的意义

Kisilevsky, Robert; Szarek, Walter A; Ancsin, John B; Elimova, Elena; Marone, Sandra; Bhat, Shridhar; Berkin, Ali