日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Hydrogel-Encapsulated Biofilm Inhibitors Abrogate the Cariogenic Activity of Streptococcus mutans

水凝胶包裹的生物膜抑制剂可消除变形链球菌的致龋活性

Ahirwar, Parmanand; Kozlovskaya, Veronika; Nijampatnam, Bhavitavya; Rojas, Edwin M; Pukkanasut, Piyasuda; Inman, Daniel; Dolmat, Maksim; Law, Anna C; Schormann, Norbert; Deivanayagam, Champion; Harber, Gregory J; Michalek, Suzanne M; Wu, Hui; Kharlampieva, Eugenia; Velu, Sadanandan E

Structural studies of antitumor compounds that target the RING domain of MDM2

靶向MDM2 RING结构域的抗肿瘤化合物的结构研究

Terrell, James Ross; Tang, Sijia; Faniyi, Oluwafoyinsola Omobodunde; Jeong, In Ho; Yin, Jun; Nijampatnam, Bhavitavya; Velu, Sadanandan E; Wang, Wei; Zhang, Ruiwen; Luo, Ming

Discovery of Potent Inhibitors of Streptococcus mutans Biofilm with Antivirulence Activity

发现具有抗毒力活性的强效变形链球菌生物膜抑制剂

Nijampatnam, Bhavitavya; Ahirwar, Parmanand; Pukkanasut, Piyasuda; Womack, Holly; Casals, Luke; Zhang, Hua; Cai, Xia; Michalek, Suzanne M; Wu, Hui; Velu, Sadanandan E

MDM2-NFAT1 dual inhibitor, MA242: Effective against hepatocellular carcinoma, independent of p53

MDM2-NFAT1双重抑制剂MA242:对肝细胞癌有效,且不依赖于p53

Wang, Wei; Cheng, Jian-Wen; Qin, Jiang-Jiang; Hu, Bo; Li, Xin; Nijampatnam, Bhavitavya; Velu, Sadanandan E; Fan, Jia; Yang, Xin-Rong; Zhang, Ruiwen

Discovery and Characterization of Dual Inhibitors of MDM2 and NFAT1 for Pancreatic Cancer Therapy

用于胰腺癌治疗的 MDM2 和 NFAT1 双重抑制剂的发现和表征

Wei Wang #, Jiang-Jiang Qin #, Sukesh Voruganti, Bhavitavya Nijampatnam, Sadanandan E Velu, Ke-He Ruan, Ming Hu, Jianwei Zhou, Ruiwen Zhang

Highly efficient delivery of potent anticancer iminoquinone derivative by multilayer hydrogel cubes

利用多层水凝胶立方体高效递送强效抗癌亚氨基醌衍生物

Xue, Bing; Wang, Wei; Qin, Jiang-Jiang; Nijampatnam, Bhavitavya; Murugesan, Srinivasan; Kozlovskaya, Veronika; Zhang, Ruiwen; Velu, Sadanandan E; Kharlampieva, Eugenia

Structure-Based Discovery of Small Molecule Inhibitors of Cariogenic Virulence

基于结构的龋齿致病性小分子抑制剂的发现

Zhang, Qiong; Nijampatnam, Bhavitavya; Hua, Zhang; Nguyen, Thao; Zou, Jing; Cai, Xia; Michalek, Suzanne M; Velu, Sadanandan E; Wu, Hui

Mitochondrial thiol modification by a targeted electrophile inhibits metabolism in breast adenocarcinoma cells by inhibiting enzyme activity and protein levels

靶向亲电试剂对线粒体硫醇的修饰通过抑制酶活性和蛋白质水平来抑制乳腺腺癌细胞的代谢

M Ryan Smith, Praveen K Vayalil, Fen Zhou, Gloria A Benavides, Reena R Beggs, Hafez Golzarian, Bhavitavya Nijampatnam, Patsy G Oliver, Robin A J Smith, Michael P Murphy, Sadanandan E Velu, Aimee Landar

Cyanobacterial Metabolite Calothrixins: Recent Advances in Synthesis and Biological Evaluation

蓝藻代谢产物卡洛丝菌素:合成和生物学评价的最新进展

Xu, Su; Nijampatnam, Bhavitavya; Dutta, Shilpa; Velu, Sadanandan E

Hydroxychalcone inhibitors of Streptococcus mutans glucosyl transferases and biofilms as potential anticaries agents

羟基查尔酮类化合物可抑制变形链球菌葡萄糖基转移酶和生物膜,作为潜在的抗龋药物

Nijampatnam, Bhavitavya; Casals, Luke; Zheng, Ruowen; Wu, Hui; Velu, Sadanandan E