日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

MRAP2 modifies the signaling and oligomerization state of the melanocortin-4 receptor.

MRAP2 改变黑皮质素-4 受体的信号传导和寡聚化状态

Sohail Iqra, Laurin Suli-Anne, Kleinau Gunnar, Chunilal Vidicha, Morton Andrew, Brenlla Alfonso, Kagiali Zeynep Cansu Uretmen, Blouin Marie-José, Tello Javier A, Beck-Sickinger Annette G, Lohse Martin J, Scheerer Patrick, Bouvier Michel, McCormick Peter, Annibale Paolo, Biebermann Heike

A Setmelanotide-like Effect at MC4R Is Achieved by MC4R Dimer Separation

通过MC4R二聚体分离实现类似塞美拉诺肽在MC4R上的作用

Reininghaus, Nanina; Paisdzior, Sarah; Höpfner, Friederike; Jyrch, Sabine; Cetindag, Cigdem; Scheerer, Patrick; Kühnen, Peter; Biebermann, Heike

Evaluation of Pharmacological Rescue of Melanocortin-4 Receptor Nonsense Mutations by Aminoglycoside

氨基糖苷类药物对黑皮质素-4受体无义突变的药理学挽救作用评价

Höpfner, Friederike; Paisdzior, Sarah; Reininghaus, Nanina; Sohail, Iqra; Scheerer, Patrick; Annibale, Paolo; Biebermann, Heike; Kühnen, Peter

A New Mechanism in THRA Resistance: The First Disease-Associated Variant Leading to an Increased Inhibitory Function of THRA2

THRA 耐药性的新机制:首个导致 THRA2 抑制功能增强的疾病相关变异

Paisdzior, Sarah; Knierim, Ellen; Kleinau, Gunnar; Biebermann, Heike; Krude, Heiko; Straussberg, Rachel; Schuelke, Markus

Correction: Ascorbate-induced oxidative stress mediates TRP channel activation and cytotoxicity in human etoposide-sensitive and -resistant retinoblastoma cells

更正:抗坏血酸诱导的氧化应激介导人依托泊苷敏感和耐药视网膜母细胞瘤细胞中TRP通道的激活和细胞毒性

Oronowicz, Jakub; Reinhard, Jacqueline; Reinach, Peter Sol; Ludwiczak, Szymon; Luo, Huan; Salem, Marah Hussain Omar Ba; Kraemer, Miriam Monika; Biebermann, Heike; Kakkassery, Vinodh; Mergler, Stefan

Differential Signaling Profiles of MC4R Mutations with Three Different Ligands

MC4R突变体与三种不同配体的差异信号传导谱

Paisdzior, Sarah; Dimitriou, Ioanna Maria; Schöpe, Paul Curtis; Annibale, Paolo; Scheerer, Patrick; Krude, Heiko; Lohse, Martin J; Biebermann, Heike; Kühnen, Peter

N- and O-Acetylated 3-Iodothyronamines Have No Metabolic or Thermogenic Effects in Male Mice

N-和O-乙酰化的3-碘甲状腺胺对雄性小鼠没有代谢或产热作用

Gachkar, Sogol; Oelkrug, Rebecca; Herrmann, Beate; Scanlan, Thomas S; Sun, Qian; Biebermann, Heike; Hoefig, Carolin S; Schomburg, Lutz; Mittag, Jens

A New Multisystem Disorder Caused by the Gαs Mutation p.F376V

由 Gαs 基因突变 p.F376V 引起的一种新的多系统疾病

Biebermann, Heike; Kleinau, Gunnar; Schnabel, Dirk; Bockenhauer, Detlef; Wilson, Louise C; Tully, Ian; Kiff, Sarah; Scheerer, Patrick; Reyes, Monica; Paisdzior, Sarah; Gregory, John W; Allgrove, Jeremy; Krude, Heiko; Mannstadt, Michael; Gardella, Thomas J; Dattani, Mehul; Jüppner, Harald; Grüters, Annette

Signal Transduction and Pathogenic Modifications at the Melanocortin-4 Receptor: A Structural Perspective

黑皮质素-4受体的信号转导和致病修饰:结构视角

Heyder, Nicolas; Kleinau, Gunnar; Szczepek, Michal; Kwiatkowski, Dennis; Speck, David; Soletto, Lucia; Cerdá-Reverter, José Miguel; Krude, Heiko; Kühnen, Peter; Biebermann, Heike; Scheerer, Patrick

Evidence of G-protein-coupled receptor and substrate transporter heteromerization at a single molecule level

单分子水平上G蛋白偶联受体和底物转运蛋白异源二聚化的证据

Fischer, Jana; Kleinau, Gunnar; Rutz, Claudia; Zwanziger, Denise; Khajavi, Noushafarin; Müller, Anne; Rehders, Maren; Brix, Klaudia; Worth, Catherine L; Führer, Dagmar; Krude, Heiko; Wiesner, Burkhard; Schülein, Ralf; Biebermann, Heike