Preclinical pharmacology of alogabat: a novel GABA(A)-α5 positive allosteric modulator targeting neurodevelopmental disorders with impaired GABA(A) signaling
alogabat 的临床前药理学研究:一种新型 GABA(A)-α5 正向变构调节剂,靶向治疗 GABA(A) 信号传导受损的神经发育障碍
期刊:Frontiers in Pharmacology
影响因子:4.8
doi:10.3389/fphar.2025.1626078
Cecere, Giuseppe; Ballard, Theresa M; Knoflach, Frederic; Honer, Michael; Hipp, Joerg F; Garces, Pilar; Mueggler, Thomas; Künnecke, Basil; Bruns, Andreas; Prinssen, Eric P; Schoenenberger, Philipp; Janz, Philipp; Redondo, Roger; Biemans, Barbara; Knust, Henner; Olivares-Morales, Andrés; Brigo, Alessandro; Schulz, Jan Michael; Bertrand, Daniel; Saxe, Michael; O'Connor, Eoin C; Hernandez, Maria-Clemencia