日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Group 3 medulloblastoma transcriptional networks collapse under domain specific EP300/CBP inhibition

第 3 组髓母细胞瘤转录网络在域特异性 EP300/CBP 抑制下崩溃

Noha A M Shendy #, Melissa Bikowitz #, Logan H Sigua #, Yang Zhang, Audrey Mercier, Yousef Khashana, Stephanie Nance, Qi Liu, Ian M Delahunty, Sarah Robinson, Vanshita Goel, Matthew G Rees, Melissa A Ronan, Tingjian Wang, Mustafa Kocak, Jennifer A Roth, Yingzhe Wang, Burgess B Freeman, Brent A Orr, 

A yeast-based system to study SARS-CoV-2 Mpro structure and to identify nirmatrelvir resistant mutations

一种基于酵母的系统,用于研究SARS-CoV-2 Mpro结构并鉴定尼尔马特雷韦耐药突变

Ou, Jin; Lewandowski, Eric M; Hu, Yanmei; Lipinski, Austin A; Aljasser, Ali; Colon-Ascanio, Mariliz; Morgan, Ryan T; Jacobs, Lian M C; Zhang, Xiujun; Bikowitz, Melissa J; Langlais, Paul R; Tan, Haozhou; Wang, Jun; Chen, Yu; Choy, John S

A yeast-based system to study SARS-CoV-2 M pro structure and to identify nirmatrelvir resistant mutations

基于酵母的系统研究 SARS-CoV-2 M pro 结构并识别尼玛瑞韦耐药突变

Jin Ou, Eric M Lewandowski, Yanmei Hu, Austin A Lipinski, Ryan T Morgan, Lian M C Jacobs, Xiujun Zhang, Melissa J Bikowitz, Paul Langlais, Haozhou Tan, Jun Wang, Yu Chen, John S Choy

Development of Dimethylisoxazole-Attached Imidazo[1,2- a]pyridines as Potent and Selective CBP/P300 Inhibitors

二甲基异恶唑连接的咪唑并[1,2- a]吡啶作为有效和选择性 CBP/P300 抑制剂的开发

Alex Muthengi, Virangika K Wimalasena, Hailemichael O Yosief, Melissa J Bikowitz, Logan H Sigua, Tingjian Wang, Deyao Li, Zied Gaieb, Gagan Dhawan, Shuai Liu, Jon Erickson, Rommie E Amaro, Ernst Schönbrunn, Jun Qi, Wei Zhang

Differential BET Bromodomain Inhibition by Dihydropteridinone and Pyrimidodiazepinone Kinase Inhibitors

二氢蝶啶酮和嘧啶二氮杂卓酮激酶抑制剂对 BET 溴结构域的差异抑制

Rezaul Md Karim, Melissa J Bikowitz, Alice Chan, Jin-Yi Zhu, Dylan Grassie, Andreas Becker, Norbert Berndt, Steven Gunawan, Nicholas J Lawrence, Ernst Schönbrunn