日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

An Imidazo[2,1-b][1,3,4]thiadiazole Derivative Inhibits the Virulence Factor α-Hemolysin by Blocking the Pullout of Its Stem Domain

一种咪唑并[2,1-b][1,3,4]噻二唑衍生物通过阻断α-溶血素茎区结构域的拉出来抑制该毒力因子。

Korotkov, Vadim S; Lukat, Peer; Di Lucrezia, Raffaella; Shekhar, Aditya; Degenhart, Carsten; Diestel, Randi; Bilitewski, Ursula; Dinkel, Klaus; Blankenfeldt, Wulf; Brönstrup, Mark

Newly identified properties of known pharmaceuticals and myxobacterial small molecules revealed by screening for autophagy modulators

通过筛选自噬调节剂,揭示了已知药物和粘细菌小分子的新特性

Fichtner, Janine; Beer, Yan Yan; Ramm, H G Mauricio; Mühlen, Sabrina; Surup, Frank; Herrmann, Jennifer; Meister, Toni Luise; Pfaender, Stephanie; Bilitewski, Ursula; Brönstrup, Mark; Müller, Rolf; Wirth, Manfred; Eskelinen, Eeva-Liisa; Schmitz, Ingo

Predicting Antimicrobial Class Specificity of Small Molecules Using Machine Learning

利用机器学习预测小分子抗菌药物的类别特异性

Gadiya, Yojana; Genilloud, Olga; Bilitewski, Ursula; Brönstrup, Mark; von Berlin, Leonie; Attwood, Marie; Gribbon, Philip; Zaliani, Andrea

Synthesis and Microbiological Activities of 3-Nitropyrazolo-[1,5-d][1,2,4]triazin-7(6H)-ones and Derivatives

3-硝基吡唑并[1,5-d][1,2,4]三嗪-7(6H)-酮及其衍生物的合成和微生物活性

Zapol'skii, Viktor A; Munoz Castillo, Diana C; Pawletta, Brigitte; Bilitewski, Ursula; Gjikaj, Mimoza; Brüdigam, Christoff; Kaufmann, Dieter E

Total Synthesis of Tosyl-Samroiyotmycin A and Its Biological Profiling

托西里-萨姆罗伊约霉素A的全合成及其生物活性分析

Kolb, Benedikt; Schmid, Fabian; Weng, Jessica; Altevogt, Luca; Pereira Rebelo, Ruben; Wank, Bianca; Baro, Angelika; Zens, Anna; Shekhar, Aditya; Bilitewski, Ursula; Sax, Sibylle; Wittlin, Sergio; Taylor, Dale; Müller, Rudolf; Laschat, Sabine

Peptide microarrays coupled to machine learning reveal individual epitopes from human antibody responses with neutralizing capabilities against SARS-CoV-2

肽微阵列与机器学习相结合,揭示了具有中和 SARS-CoV-2 能力的人类抗体反应的单个表位

Sven-Kevin Hotop, Susanne Reimering, Aditya Shekhar, Ehsaneddin Asgari, Ulrike Beutling, Christine Dahlke, Anahita Fathi, Fawad Khan, Marc Lütgehetmann, Rico Ballmann, Andreas Gerstner, Werner Tegge, Luka Cicin-Sain, Ursula Bilitewski, Alice C McHardy, Mark Brönstrup

Reprogramming of Amino Acid Metabolism Differs between Community-Acquired Pneumonia and Infection-Associated Exacerbation of Chronic Obstructive Pulmonary Disease

社区获得性肺炎和慢性阻塞性肺疾病感染相关性急性加重患者的氨基酸代谢重编程存在差异

Arshad, Haroon; Siokis, Anastasios; Franke, Raimo; Habib, Aamna; Alfonso, Juan Carlos López; Poliakova, Yuliya; Lücke, Eva; Michaelis, Katina; Brönstrup, Mark; Meyer-Hermann, Michael; Bilitewski, Ursula; Vila, Jordi; Abel, Laurent; Illig, Thomas; Schreiber, Jens; Pessler, Frank

Identification of Antimotilins, Novel Inhibitors of Helicobacter pylori Flagellar Motility That Inhibit Stomach Colonization in a Mouse Model

鉴定抗胃动素,一种抑制小鼠模型中胃定植的幽门螺杆菌鞭毛运动的新型抑制剂

Sebastian Suerbaum #, Nina Coombs, Lubna Patel, Dimitri Pscheniza, Katharina Rox, Christine Falk, Achim D Gruber, Olivia Kershaw, Patrick Chhatwal, Mark Brönstrup, Ursula Bilitewski, Christine Josenhans #

Chemistry of polyhalogenated nitrobutadienes, 17: Efficient synthesis of persubstituted chloroquinolinyl-1H-pyrazoles and evaluation of their antimalarial, anti-SARS-CoV-2, antibacterial, and cytotoxic activities

多卤代硝基丁二烯的化学,17:全取代氯喹啉基-1H-吡唑的高效合成及其抗疟疾、抗SARS-CoV-2、抗菌和细胞毒活性评价

Zapol'skii, Viktor A; Berneburg, Isabell; Bilitewski, Ursula; Dillenberger, Melissa; Becker, Katja; Jungwirth, Stefan; Shekhar, Aditya; Krueger, Bastian; Kaufmann, Dieter E

Identification of Translocation Inhibitors Targeting the Type III Secretion System of Enteropathogenic Escherichia coli

鉴定靶向肠致病性大肠杆菌III型分泌系统的转位抑制剂

Mühlen, Sabrina; Zapol'skii, Viktor A; Bilitewski, Ursula; Dersch, Petra