日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

An Imidazo[2,1-b][1,3,4]thiadiazole Derivative Inhibits the Virulence Factor α-Hemolysin by Blocking the Pullout of Its Stem Domain

一种咪唑并[2,1-b][1,3,4]噻二唑衍生物通过阻断α-溶血素茎区结构域的拉出来抑制该毒力因子。

Korotkov, Vadim S; Lukat, Peer; Di Lucrezia, Raffaella; Shekhar, Aditya; Degenhart, Carsten; Diestel, Randi; Bilitewski, Ursula; Dinkel, Klaus; Blankenfeldt, Wulf; Brönstrup, Mark

Newly identified properties of known pharmaceuticals and myxobacterial small molecules revealed by screening for autophagy modulators

通过筛选自噬调节剂,揭示了已知药物和粘细菌小分子的新特性

Fichtner, Janine; Beer, Yan Yan; Ramm, H G Mauricio; Mühlen, Sabrina; Surup, Frank; Herrmann, Jennifer; Meister, Toni Luise; Pfaender, Stephanie; Bilitewski, Ursula; Brönstrup, Mark; Müller, Rolf; Wirth, Manfred; Eskelinen, Eeva-Liisa; Schmitz, Ingo

Predicting Antimicrobial Class Specificity of Small Molecules Using Machine Learning

利用机器学习预测小分子抗菌药物的类别特异性

Gadiya, Yojana; Genilloud, Olga; Bilitewski, Ursula; Brönstrup, Mark; von Berlin, Leonie; Attwood, Marie; Gribbon, Philip; Zaliani, Andrea

Synthesis and Microbiological Activities of 3-Nitropyrazolo-[1,5-d][1,2,4]triazin-7(6H)-ones and Derivatives

3-硝基吡唑并[1,5-d][1,2,4]三嗪-7(6H)-酮及其衍生物的合成和微生物活性

Zapol'skii, Viktor A; Munoz Castillo, Diana C; Pawletta, Brigitte; Bilitewski, Ursula; Gjikaj, Mimoza; Brüdigam, Christoff; Kaufmann, Dieter E

Total Synthesis of Tosyl-Samroiyotmycin A and Its Biological Profiling

托西里-萨姆罗伊约霉素A的全合成及其生物活性分析

Kolb, Benedikt; Schmid, Fabian; Weng, Jessica; Altevogt, Luca; Pereira Rebelo, Ruben; Wank, Bianca; Baro, Angelika; Zens, Anna; Shekhar, Aditya; Bilitewski, Ursula; Sax, Sibylle; Wittlin, Sergio; Taylor, Dale; Müller, Rudolf; Laschat, Sabine

Reprogramming of Amino Acid Metabolism Differs between Community-Acquired Pneumonia and Infection-Associated Exacerbation of Chronic Obstructive Pulmonary Disease

社区获得性肺炎和慢性阻塞性肺疾病感染相关性急性加重患者的氨基酸代谢重编程存在差异

Arshad, Haroon; Siokis, Anastasios; Franke, Raimo; Habib, Aamna; Alfonso, Juan Carlos López; Poliakova, Yuliya; Lücke, Eva; Michaelis, Katina; Brönstrup, Mark; Meyer-Hermann, Michael; Bilitewski, Ursula; Vila, Jordi; Abel, Laurent; Illig, Thomas; Schreiber, Jens; Pessler, Frank

Chemistry of polyhalogenated nitrobutadienes, 17: Efficient synthesis of persubstituted chloroquinolinyl-1H-pyrazoles and evaluation of their antimalarial, anti-SARS-CoV-2, antibacterial, and cytotoxic activities

多卤代硝基丁二烯的化学,17:全取代氯喹啉基-1H-吡唑的高效合成及其抗疟疾、抗SARS-CoV-2、抗菌和细胞毒活性评价

Zapol'skii, Viktor A; Berneburg, Isabell; Bilitewski, Ursula; Dillenberger, Melissa; Becker, Katja; Jungwirth, Stefan; Shekhar, Aditya; Krueger, Bastian; Kaufmann, Dieter E

Identification of Translocation Inhibitors Targeting the Type III Secretion System of Enteropathogenic Escherichia coli

鉴定靶向肠致病性大肠杆菌III型分泌系统的转位抑制剂

Mühlen, Sabrina; Zapol'skii, Viktor A; Bilitewski, Ursula; Dersch, Petra

Inhibition of Type IV Secretion Activity and Growth of Helicobacter pylori by Cisplatin and Other Platinum Complexes.

顺铂和其他铂配合物对幽门螺杆菌IV型分泌活性和生长的抑制作用

Lettl Clara, Schindele Franziska, Testolin Giambattista, Bär Alexander, Rehm Tobias, Brönstrup Mark, Schobert Rainer, Bilitewski Ursula, Haas Rainer, Fischer Wolfgang

Polyhalonitrobutadienes as Versatile Building Blocks for the Biotargeted Synthesis of Substituted N-Heterocyclic Compounds

多卤代硝基丁二烯作为生物靶向合成取代N-杂环化合物的多功能结构单元

Zapol'skii, Viktor A; Bilitewski, Ursula; Kupiec, Sören R; Ramming, Isabell; Kaufmann, Dieter E