Novel small molecule analogs for advancing apelin receptor antagonism with enhanced plasma and microsomal stability
新型小分子类似物可增强apelin受体拮抗作用,并提高血浆和微粒体稳定性
期刊:Bioorganic & Medicinal Chemistry Letters
影响因子:2.2
doi:10.1016/j.bmcl.2025.130367
Bist, Ganesh; Elsheikh, Ahmed; Kim, Sewon; Huang, Ruea-Yea; Ruszaj, Donna; Woo, Sukyung; You, Youngjae